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SK&F-105517-D

Phase 1

Heart Failure, Congestive | Small molecule | Cardiovascular |GSK plc|Last Updated: Aug 2, 2017

Success Probability

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Market & Valuation

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Trial Design

RandomizedCONTROLLED
Total Trials1
Total Enrollment41

FDA Designations

No designations recorded

Clinical trial landscape

SK&F-105517-D · 1 trial · 1 indication

Phase 1 1
NCT00742508A Phase I/II Clinical Study of SK&F-105517-D in Japanese Patients With Chronic Heart FailureHeart Failure, Congestive
COMPLETED41 Analytics
PHASE1COMPLETED
A Phase I/II Clinical Study of SK&F-105517-D in Japanese Patients With Chronic Heart Failure
Heart Failure, CongestiveUnlock trial analytics

Study Endpoints

Primary Endpoints

Number of Participants With Adverse Events by Severity From Week 0 Through Week 8 (CRV-IR) or Week 14 (SK&F-105517-D)
Treatment Period from Week 0 (Baseline) to Week 8 and 1-week Follow-up Period (Week 9) for CRV-IR; Treatment Period from Week 0 (Baseline) to Week 14 and 1-week Follow-up Period (Week 15) for SK&F-105517-D

Drug-related adverse events (AEs) were defined as AEs that were judged to have a relationship with the investigational product by the investigator (or subinvestigator) with the use of clinical judgment and the Clinical Investigator Brochure to determine the relationship. Refer to adverse event information for type and frequency of adverse events.

Mean Change From Baseline in Albumin and Total Protein at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Alkaline Phosphatase, Alanine Aminotransferase, Aspartate Aminotransferase, Creatine Kinase, and Gamma Glutamyl Transferase at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value

Mean Change From Baseline in Amylase at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value

Mean Change From Baseline in Total Bilirubin, Creatinine, and Uric Acid at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value

Mean Change From Baseline in Calcium, Chloride, Glucose, Potassium, Sodium, and Urea/Blood Urea Nitrogen at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value

Mean Change From Baseline in Creatine Kinase BB Percentage, Creatine Kinase MB Percentage, and Creatine Kinase MM Percentage at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value. (BB, brain-derived; MB=cardiac muscle-derived; MM=skeletal muscle-derived.

Mean Change From Baseline in Each Type of White Blood Cell (WBC) (Basophils, Eosinophils, Lymphocytes, Monocytes, and Total Neutrophils) at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Hemoglobin and Mean Corpuscular Hemoglobin Concentration at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Hematocrit at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Platelet Count and White Blood Cell Count at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Red Blood Cell Count at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Mean Corpuscular Hemoglobin at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Mean Corpuscular Volume at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Number of Participants With the Indicated Urinalysis Dipstick Results at Baseline and Week 8
Baseline and Week 8

Dipstick test values: Negative (-), Traces (+-), +1, +2, +3. +4. Normal ranges (qualitative): protein, - or +-; glucose, - or +-; occult blood, -; ketones, -.

Mean Change From Baseline in Systolic Blood Pressure and Diastolic Blood Pressure at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Heart Rate at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Mean Change From Baseline in Weight at Week 8
Baseline and Week 8

Mean change from baseline was calculated as the Week 8 value minus the Baseline value.

Number of Participants With the Indicated Electrocardiogram Findings at Baseline and Week 8
Baseline and Week 8

There are 3 categories for electrocardiogram (ECG) findings: normal; abnormal, not clinically significant; and abnormal, clinically significant. Each of the findings was classified by the investigator according to whether it was normal. Abnormal ECGs were further classified according to whether they were felt to be clinically significant in the medical and scientific judgment of the investigator.

Cardiothoracic Ratio at Baseline and Week 8
Baseline and Week 8

Cardiothoracic ratio is a marker of the degree of heart enlargement and was measured by chest X-ray. It is shown as the ratio of the transverse diameter of the heart to the transverse diameter of the thorax, and is measured as a percentage.

Secondary Endpoints

Maximum Plasma Concentration (Cmax) and Trough Plasma Concentration (Cmin) of S-carvedilol, R-carvedilol, and M4 Active Metabolite (SB-203231) at Week 8
Week 8
Area Under the Plasma Concentration Versus Time Curve From Time Zero to 24 Hours (AUC0-24) of S-carvedilol, R-carvedilol, and M4 Active Metabolite (SB-203231) at Week 8
Week 8
Time of Maximal Plasma Concentration (Tmax) of S-carvedilol, R-carvedilol, and M4 Active Metabolite (SB-203231) at Week 8
Week 8
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
SK&F-105517-D groupEXPERIMENTALSK\&F-105517-D 10-80 mg/day
Carvedilol-IR groupOTHERCarvedilol-IR 5-20 mg/day

Interventions

NameTypeDescription
SK&F-105517-D 10 mg capsuleDRUG1 capsule once a day
Carvedilol-immediate release (IR) 2.5 mg tabletDRUG1 or 2 tablet(s) twice a day
SK&F-105517-D 20 mg capsuleDRUG1 capsule once a day
SK&F-105517-D 40 mg capsuleDRUG1 or 2 capsule(s) once a day
Carvedilol-IR 10 mg tabletDRUG1 tablet twice a day
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Eligibility Criteria

Age Range20 Years to 80 Years
SexALL
Healthy VolunteersNo
Study Sites23

Inclusion criteria: * Patients with symptomatically stable chronic heart failure (CHF) based on ischemic heart disease or dilated cardiomyopathy * Patients who are maintained on basic heart failure therapy with angiotensin converting enzyme (ACE) inhibitors or angiotensin II receptor blocker (ARB) ...

Countries:Japan
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Frequently asked questions about SK&F-105517-D

What is SK&F-105517-D used for?

SK&F-105517-D is an investigational small molecule being studied for the treatment of congestive heart failure. It has been evaluated in a clinical trial involving Japanese patients with chronic heart failure. The drug is in Phase 1 of clinical development and is not yet approved for any use.

Who makes SK&F-105517-D?

SK&F-105517-D is being developed by GSK plc, a global pharmaceutical company listed on the stock exchange under the ticker GSK. The company conducted a clinical trial of this drug in Japan for the treatment of congestive heart failure.

What phase is SK&F-105517-D in?

SK&F-105517-D is in Phase 1 of clinical development. It has completed one Phase 1/II clinical trial in Japan, which enrolled 41 patients with chronic heart failure. The drug remains investigational and has not received regulatory approval.

What clinical trials is SK&F-105517-D in?

SK&F-105517-D has been studied in one completed clinical trial, registered as NCT00742508. This was a Phase I/II study in Japanese patients with chronic heart failure, enrolling 41 participants. The trial was controlled and randomized, though not double-blind, and included both male and female patients aged 20 years and older.

Is SK&F-105517-D the same as any other drug?

SK&F-105517-D is the specific drug name used in clinical development. No alternative names have been reported for this compound. It is a small molecule being investigated for congestive heart failure, and no other designations have been associated with it in the available information.