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SB-756050 immediate release

Phase 1

Diabetes Mellitus, Type 2 | Small molecule | Metabolic |GSK plc|Last Updated: Sep 6, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment36
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00607906First-Time-in-Humans Study to Assess Safety, Pharmacokinetics & Pharmacodynamics of SB756050PHASE1 COMPLETED 36Nov 16, 2007Mar 10, 2008Sep 6, 20171 United States
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Study Endpoints
Primary Endpoints
adverse events:
each visit
clinical laboratory:
day -1, day 2 each period
electrocardiogram (ECG):
day 1 each period
vital signs assessments:
day -1, day 1 each period
Secondary Endpoints
plasma drug concentrations:
Day 1 each dosing level
plasma blood sugar & other parameter concentrations:
Day 1 Period 4 following meal
Correlation between drug concentrations & blood sugar levels:
day 1 period 4
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Study Design & Arms
AllocationRANDOMIZED
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Subjects receiving treatment in cohort A1EXPERIMENTALEligible subjects will receive oral immediate release capsules of SB-756050 with doses of 5 milligrams, 15 milligrams, 50 milligrams, or 100 milligrams.
Subjects receiving treatment in cohort A2EXPERIMENTALEligible subjects will receive oral immediate release capsules of SB-756050 with doses of 100 milligrams, 200 milligrams, 300 milligrams, or 400 milligrams.
Subjects receiving treatment in cohort A3EXPERIMENTALEligible subjects will receive oral immediate release capsules of SB-756050 with a dose of 150 milligrams. Subjects will also receive oral modified release capsules of SB-756050 with doses of 150 milligrams, 300 milligrams, or 400 milligrams.
Subjects receiving treatment in cohort A4EXPERIMENTALEligible subjects will receive SB-756050 in this additional cohort.
Subjects receiving treatment in cohort B1EXPERIMENTALEligible subjects will receive oral modified release capsules of SB-756050 with doses of 50 milligrams, 150 milligrams or 400 milligrams. Subjects will also receive immediate release oral capsules of SB-756050 with a dose of 150 milligrams.
Interventions
NameTypeDescription
SB-756050 immediate release capsuleDRUGSB-756050 immediate release capsules will be size 0, white, opaque capsules with no identifying markings, containing white to off-white drug layered pellets. Each capsule will contain 5, 25 or 100 milligrams of SB-756050.
SB-756050 modified release capsuleDRUGSB-756050 modified release capsules will be size 0, white, opaque capsules with no identifying markings, containing white to off-white enteric coated drug layered pellets. Each capsule will contain either 25or 100 milligrams of SB-756050.
PlaceboDRUGSubjects will also receive placebo capsules.
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Eligibility Criteria
Age Range18 Years — 60 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: Healthy Subjects * Healthy male or female subject as determined by a responsible physician, based on a medical evaluation including history, physical examination, vitals signs, laboratory tests, and cardiac monitoring. * Female subjects must be of non-childbearing potential inc...

Countries:United States
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