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Ronacaleret

Phase 1

Bone Marrow Transplantation | Small molecule | Hematology |GSK plc|Last Updated: Jun 20, 2017

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment39

FDA Designations

No designations recorded

Clinical trial landscape

Ronacaleret · 3 trials · 3 indications

Phase 1 3
NCT01802892Study in Healthy Volunteers, to Evaluate the Safety, Efficacy and Dose Responses of SB-751689 (Ronacaleret)Transplantation, Stem Cell
COMPLETED24 Analytics
NCT01466335An Adaptive Phase I Study to Evaluate the Safety, Efficacy and Dose Responses of Ronacaleret in Healthy Human VolunteersBone Marrow Transplantation
COMPLETED39 Analytics
NCT00651534To Estimate Relative Bioavailability of 5 Formulations of Ronacaleret Given to Healthy Postmenopausal FemalesOsteoporosis
COMPLETED32 Analytics
PHASE1COMPLETED
Study in Healthy Volunteers, to Evaluate the Safety, Efficacy and Dose Responses of SB-751689 (Ronacaleret)
Transplantation, Stem CellUnlock trial analytics
PHASE1COMPLETED
An Adaptive Phase I Study to Evaluate the Safety, Efficacy and Dose Responses of Ronacaleret in Healthy Human Volunteers
Bone Marrow TransplantationUnlock trial analytics
PHASE1COMPLETED
To Estimate Relative Bioavailability of 5 Formulations of Ronacaleret Given to Healthy Postmenopausal Females
OsteoporosisUnlock trial analytics

Study Endpoints

Primary Endpoints

Mean change from baseline in CD34+ cell counts
Baseline and upto Day 14

The mean fold change from baseline in the number of circulating CD34+ cells for all treatment arms will be assessed. Samples will be collected at screening, Day 4 and Day 5 (2 hrs post ronacaleret dose), Day 6 (12 hrs and 14 and 16 hrs post plerixafor dose) and Day 14

assess the mean fold increase in the number of peripheral CD34+ cells, at total daily doses ranging from 100mg to 400mgs over 1 to 28 days
1-28 days

Secondary Endpoints

Spontaneous AE reporting
Up to 14 days
Clinical laboratory safety data
Up to 14 days
Measure of vital signs to access safety and tolerability
Up to 14 days
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Ronacaleret 100 mgEXPERIMENTALSubjects will receive ronacaleret (100 mg once daily) for 5 consecutive days, given in conjunction with a single dose of plerixafor (0.24 mg/kg) SC on the evening of Day 5.
Ronacaleret 400 mgEXPERIMENTALSubjects will receive ronacaleret (400 mg once daily) for 5 consecutive days, given in conjunction with a single dose of plerixafor (0.24 mg/kg) SC on the evening of Day 5.
Ronacaleret 100mg once dailyEXPERIMENTAL1 x 100mg oral tablet
Ronacaleret 100mg twice dailyEXPERIMENTAL1 x 100mg oral tablet twice daily
Ronacaleret 200mg once dailyEXPERIMENTAL2 x 100mg oral tablet
Ronacaleret 200mg twice dailyEXPERIMENTAL2 x 100mg tablets twice daily
Ronacaleret 400mg once dailyEXPERIMENTAL4 x 100mg tablets
PlaceboPLACEBO_COMPARATORMatching number of identical placebo tablets

Interventions

NameTypeDescription
Ronacaleret 100 mgDRUGSubjects in the Ronacaleret 100 mg group received one tablet orally of ronacaleret 100 mg for 5 consecutive days.
Ronacaleret 400 mgDRUGSubjects in the Ronacaleret 400 mg group received four tablets orally of ronacaleret 100 mg daily for 5 consecutive days.
PlerixaforDRUGSubjects in each group received a single dose of plerixafor (0.24mg/kg) SC on the evening of the Day 5 dosing approximately 12 hours before collection of CD34+ cells on day 6.
Ronacaleret (100mg tablet)DRUG100mg tablet
PlaceboDRUGmatching placebo tablet
RonacaleretDRUG -
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * A male or female between 18 and 65 years of age (inclusive). * Healthy as determined by a physician, based on a medical evaluation and with an estimated Glomerular Filtration Rate (GFR) of \>=60 mL/min /1.73 m\^2 using the four variable Modification of Diet in Renal Disease (M...

Countries:United States
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Frequently asked questions about Ronacaleret

What is Ronacaleret used for?

Ronacaleret is an investigational small molecule being studied for osteoporosis, transplantation, stem cell, and bone marrow transplantation. It is being developed by GSK plc (GSK) and is currently in Phase 1 clinical development. Ronacaleret is not approved by the FDA and remains under investigation.

What does Ronacaleret target?

Ronacaleret is a small molecule developed by GSK plc (GSK). Its specific molecular target has not been disclosed in available information. The drug is being investigated for potential use in osteoporosis and transplantation-related conditions, but its mechanism of action is not publicly detailed.

Who makes Ronacaleret?

Ronacaleret is being developed by GSK plc, a global pharmaceutical company traded on the New York Stock Exchange under the ticker GSK. The drug is currently in Phase 1 clinical trials and is not yet approved for any indication.

What phase is Ronacaleret in?

Ronacaleret is in Phase 1 clinical development. It has completed three Phase 1 trials, all of which are finished. The drug remains investigational and has not received FDA approval. GSK plc (GSK) is the developer of Ronacaleret.

What clinical trials is Ronacaleret in?

Ronacaleret has completed three Phase 1 clinical trials: NCT00651534, NCT01466335, and NCT01802892. These trials evaluated the drug in healthy volunteers for conditions including osteoporosis, bone marrow transplantation, and stem cell transplantation. All trials are completed, with no active trials currently ongoing.

Is Ronacaleret the same as SB-751689?

Yes, Ronacaleret is also known as SB-751689. The clinical trial NCT01802892, titled 'Study in Healthy Volunteers, to Evaluate the Safety, Efficacy and Dose Responses of SB-751689 (Ronacaleret)', confirms that SB-751689 is an alternative name for Ronacaleret.