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Raltegravir

Phase 1

Infection, Human Immunodeficiency Virus | Small molecule | Other |GSK plc|Last Updated: Sep 11, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment15
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01101893A Drug Interaction Study Evaluating GSK2248761 and Raltegravir Pharmacokinetics in Healthy Adult SubjectsPHASE1 COMPLETED 15Apr 1, 2010Jun 1, 2010Sep 11, 20171 United States
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Study Endpoints
Primary Endpoints
Plasma raltegravir steady-state CL/F, AUC(0-tau), Cmax, tmax, Ctau, and Cmin following administration of raltegravir 400mg q12h for 5 days and following co-administration with GSK2248761 200mg q24h for 5 days.
5 days
Plasma GSK2248761 steady state PK parameters, including CL/F, AUC(0-tau), Cmax, tmax, Ctau, & Cmin following administration of GSK2248761 200mg q24h for 5 days & following co-administration of raltegravir 400 mg q12h & GSK2248761 200 mg q24h for 5 days
5 days
Secondary Endpoints
Safety and tolerability parameters, including adverse event, concurrent medication, clinical laboratory, ECG, and vital signs assessments
approximately 34 days
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeOTHER
Treatment Arms
ArmTypeDescription
Period 1EXPERIMENTALIn period 1 all subjects will receive Raltegravir 400mg q12h from Day 1 to Day 5
Period 2EXPERIMENTALIn period 2 all subjects will receive GSK2248761 200mg q24h from Day 1 to Day 5.
Period 3EXPERIMENTALDay 1 of Period 3 will be the day after Day 5 of Period 2. Subjects will receive GSK2248761 200mg q24h + raltegravir 400mg q12h from Day 1 to Day 5.
Interventions
NameTypeDescription
RaltegravirDRUGraltegravir 400mg q12h x 5 days (Reference Treatment)
GSK2248761DRUGGSK2248761 200mg q24h x 5 days (Reference Treatment)
GSK2248761 + RaltegravirDRUGGSK2248761 200mg q24h + raltegravir 400mg q12h x 5 days (Test Treatment)
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Eligibility Criteria
Age Range18 Years — 50 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy as determined by a responsible and experienced physician, based on a medical evaluation including medical history, physical examination, vital signs, laboratory tests, and ECGs. A subject with a clinical abnormality or laboratory parameters outside the reference range ...

Countries:United States
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