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Ortho-Cyclen

Phase 1

Infection, Human Immunodeficiency Virus | Small molecule | Other |GSK plc|Last Updated: May 21, 2012

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDBiomarker
Total Trials1
Total Enrollment16
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01498861Drug Interaction Study Between Dolutegravir and an Oral Contraceptive Containing Norgestimate and EthinylestradiolPHASE1 COMPLETED 16Dec 1, 2011Mar 1, 2012May 21, 20121 United States
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Study Endpoints
Primary Endpoints
AUC(0-tau) of norelgestromin and ethinylestradiol after Ortho-Cyclen alone and after Ortho-Cyclen with dolutegravir
Up to 24 hours post-dose

Samples will be collected at predose and at 0.5, 1, 1.5, 2, 2.5, 3, 4, 6, 8, 10, 12, and 24 hours postdose on Days 10 and 21

Secondary Endpoints
Safety and tolerability of all treatments as assessed by vital signs, AEs, and clinical laboratory tests
Up to 8 weeks
Composite of norelgestromin pharmacokinetic parameters on Day 10 and Day 21: Cmax, Cmin, tmax, tmin and half life
Up to 24 hours post dose
Predose serum levels of luteinizing hormone and follicle stimulating hormone from Periods 1 and 2
predose on Days 1, 10, 11, 21 and 22
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelCROSSOVER
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
Run-In PeriodOTHEROrtho-Cyclen for 21 days. Only for subjects who are not already taking Ortho-Cyclen prior to the study
Sequence ABEXPERIMENTALSubjects will take Ortho-Cyclen once a day from Day 1-21 of their menstrual cycle. In addition they will take dolutegravir 50 mg twice a day from Days 1-10 and placebo twice a day from Day 12-21
Sequence BAEXPERIMENTALSubjects will take Ortho-Cyclen once a day from Day 1-21 of their menstrual cycle. In addition they will take placebo twice a day from Days 1-10 and dolutegravir 50 mg twice a day from Day 12-21
Interventions
NameTypeDescription
Ortho-CyclenDRUGOrtho-cyclen is an oral contraceptive.
DolutegravirDRUGDolutegravir is an experimental HIV drug
PlaceboDRUGPlacebo is a tablet with no drug in it
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Eligibility Criteria
Age Range18 Years — 40 Years
SexFEMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Alanine aminotransferase (ALT), alkaline phosphatase and bilirubin greater than or equal to 1.5 times the upper limit of normal (ULN) * Healthy female subjects, as determined by a responsible and experienced physician, based on a medical evaluation including medical history, p...

Countries:United States
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