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GSK586529

Phase 1

Depressive Disorder and Anxiety Disorders | Small molecule | Psychiatry |GSK plc|Last Updated: Aug 22, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment21
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00703547A First Time in Human Study of GSK586529 in Healthy VolunteersPHASE1 COMPLETED 21Jan 28, 2008Apr 11, 2008Aug 22, 20171 United Kingdom
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Study Endpoints
Primary Endpoints
Pharmacokinetics
Pre-dose, 30 minutes, 1, 2, 3, 4, 6, 8, 12, 24, 36, 48, 72 and 96 hours post-dose
Secondary Endpoints
Blood levels of GSK586529 to determine pharmacokinetic parameters
Pre-dose, 30 minutes, 1, 2, 3, 4, 6, 8, 12, 24, 36, 48, 72 and 96 hours post-dose
Urinary recovery of GSK586529
Pre-dose, 0-6, 6-12, 12-24, 24-48, 48-72 and 72-96 hours post-dose
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Study Design & Arms
AllocationRANDOMIZED
ModelCROSSOVER
PurposePREVENTION
Treatment Arms
ArmTypeDescription
Subjects receiving treatment in cohort 1EXPERIMENTALSubjects will receive one of the following sequences; ABDF,BADF, BDAF or BDFA (A=Placebo, B= GSK586529 dose 1 (3 milligrams), D = GSK586529 dose 3, F = GSK586529 dose 5).
Subjects receiving treatment in cohort 2EXPERIMENTALSubjects will receive one of the following sequences; ACEG,CAEG, CEAG or CEGA (A = Placebo, C= GSK586529 dose 2, E = GSK586529 dose 4, G = GSK586529 dose 6)
Interventions
NameTypeDescription
GSK586529 capsulesDRUGGSK586529 will be provided as white gelatin capsule with a dose of 3 milligrams.
GSK586529 tabletsDRUGGSK586529 will be provided as a yellow film-coated tablets for oral administration at three different strengths 10 milligrams, 60 milligrams and 120 milligrams.
PlaceboDRUGPlacebo tablets and capsules will be provided to subjects.
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Eligibility Criteria
Age Range18 Years — 45 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy males aged 18-45 years, inclusive. * Healthy subjects, defined as individuals who are free from clinically significant illness or disease as determined by their (and familial) medical and psychiatric history, physical examination, laboratory studies, and other tests. *...

Countries:United Kingdom
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