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GSK461364

Phase 1

Lymphoma, Non-Hodgkin | Small molecule | Oncology |GSK plc|Last Updated: Jun 26, 2017

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment41

FDA Designations

No designations recorded

Clinical trial landscape

GSK461364 · 1 trial · 1 indication

Phase 1 1
NCT00536835Study to Assess the Pharmacokinetics and Pharmacodynamics of GSK461364 in Subjects With Non-Hodgkins LymphomaLymphoma, Non-Hodgkin
COMPLETED41 Analytics
PHASE1COMPLETED
Study to Assess the Pharmacokinetics and Pharmacodynamics of GSK461364 in Subjects With Non-Hodgkins Lymphoma
Lymphoma, Non-HodgkinUnlock trial analytics

Study Endpoints

Primary Endpoints

Plasma levels for GSK461364 will be taken at:Schedule 1:Day 1, 8, 15, & 22 for Cycle 1 and Day 1, 8 & 15 for subsequent cycles.Schedule 2:Day 1, 2, 8, 9, 15, & 16 for all cycles.Schedule 3:Day 1 to 5 for all cycles.
16 Days

Secondary Endpoints

Safety will be evaluated by: - Physical exam at screen & then D1 for each cycle - 12 lead ECG & telemetry at screen & Wk 1 to 3 for Schedule 1 & 2, & Wk 1 & 2 (ECG only) for Schedule 3. - Lab tests & AE monitoring throughout the study.
16 Days
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Stage AEXPERIMENTALStage A will identify maximum tolerated doses for either Schedule 1 - GSK461364 given once weekly on Day 1, 8 and 15 every 28 days; Schedule 2 - GSK 461364 given twice weekly Days 1, 2, 8, 9, 15 and 16; Schedule 3 Daily on Day 1 to Day 15 every 21 days.
Stage BEXPERIMENTALEvaluate safety, PK, pharmacodynamic (PD) \& tumor response in expanded cohorts at the MTD for at least one schedule from Stage A.

Interventions

NameTypeDescription
GSK461364DRUGGSK461364 will be given intravenously as a 4 hour infusion in either a final volume of 500 or 1000 mLs. The starting dose for Stage A - Schedule 1 was 50 mg and doses were to be escalated as described in protocol until maximum tolerated dose established.
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites3

Inclusion Criteria: * Confirmed diagnosis of advanced solid tumor or Non-Hodgkins Lymphoma (excluding HIV-associated lymphoma) that has relapsed or is refractory to standard therapies * At least 18 years of age * Female who are of non-childbearing potential or who have a negative pregnancy test who...

Countries:United Kingdom
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Frequently asked questions about GSK461364

What is GSK461364 used for?

GSK461364 is an investigational small molecule being studied for the treatment of Non-Hodgkin lymphoma. It was evaluated in a Phase 1 clinical trial that has been completed. The drug is not approved and remains in clinical development.

Who makes GSK461364?

GSK461364 is being developed by GSK plc, a pharmaceutical company traded on the New York Stock Exchange under the ticker symbol GSK. The company conducted a Phase 1 study of the drug in subjects with Non-Hodgkin lymphoma.

What phase is GSK461364 in?

GSK461364 is in Phase 1 clinical development. A Phase 1 study of the drug in Non-Hodgkin lymphoma has been completed. The drug is investigational and has not been approved by regulatory authorities.

What clinical trials is GSK461364 in?

GSK461364 has one completed clinical trial, NCT00536835, titled 'Study to Assess the Pharmacokinetics and Pharmacodynamics of GSK461364 in Subjects With Non-Hodgkins Lymphoma.' This Phase 1 study enrolled 41 participants in the United Kingdom.

Is GSK461364 FDA approved?

GSK461364 is not FDA approved. It is an investigational drug that has completed a Phase 1 clinical trial for Non-Hodgkin lymphoma. The drug remains in clinical development and has not been authorized for commercial use.