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GSK2376497

Phase 1

Diabetes Mellitus, Type 2 | Small molecule | Metabolic |GSK plc|Last Updated: Jul 25, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment82
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01545570A Study to Determine the Safety, Tolerability, and Effects of GSK2374697 in Healthy VolunteersPHASE1 COMPLETED 82Nov 7, 2011Dec 23, 2012Jul 25, 20171 United States
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Study Endpoints
Primary Endpoints
Number of subjects with adverse events after ascending single or titrated mulitple subcutaneous doses of GSK2374697
up to 70 days post dose

Adverse events, laboratory parameters, ECGs, and vital signs

pharmacokinetic parameters of GSK2374697, after ascending single or titrated multiple subcutaneous doses, in healthy subjects
pre-dose, then 6, 12, 18, 24, 30, 36, 42, 48, 54, 60, and 66 hours after dose (this schedule is q6h through Day 3, up to just prior to Day 4). In addition, sampling continues out through Day 70, on specific days, q12h.

Pharmacokinetics parameters: AUCs, Cmax, tmax, elimination half-life (t½), lag time (tlag), apparent clearance (CL/F) and apparent volume of distribution (V/F), area under the plasma drug concentration versus time curve on Days 1 through end of study (up to 70 Days)

Secondary Endpoints
pharmacodynamic effects of GSK2374697 in healthy subjects after meal challenge
On 2 days
dose proportionality of GSK2374697
up to 70 days post dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
GSK2376497ACTIVE_COMPARATORsingle dose escalation or multiple-dose titration
0.9% sodium chloridePLACEBO_COMPARATORplacebo injection
Interventions
NameTypeDescription
GSK2376497DRUGGSK2376497 Active Comparator
0.9% sodium chlorideDRUG0.9% sodium chloride Placebo Comparator
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Eligibility Criteria
Age Range18 Years — 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy as determined by a responsible and experienced physician, based on a medical evaluation including medical history, physical examination, laboratory tests and Holter monitoring. A subject with a clinical abnormality or laboratory parameters outside the reference range f...

Countries:United States
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