Recent Updates
Recently added Catalysts

GSK2376497

Phase 1

Diabetes Mellitus, Type 2 | Small molecule | Metabolic |GSK plc|Last Updated: Jul 25, 2017

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment82

FDA Designations

No designations recorded

Clinical trial landscape

GSK2376497 · 1 trial · 1 indication

Phase 1 1
NCT01545570A Study to Determine the Safety, Tolerability, and Effects of GSK2374697 in Healthy VolunteersDiabetes Mellitus, Type 2
COMPLETED82 Analytics
PHASE1COMPLETED
A Study to Determine the Safety, Tolerability, and Effects of GSK2374697 in Healthy Volunteers
Diabetes Mellitus, Type 2Unlock trial analytics

Study Endpoints

Primary Endpoints

Number of subjects with adverse events after ascending single or titrated mulitple subcutaneous doses of GSK2374697
up to 70 days post dose

Adverse events, laboratory parameters, ECGs, and vital signs

pharmacokinetic parameters of GSK2374697, after ascending single or titrated multiple subcutaneous doses, in healthy subjects
pre-dose, then 6, 12, 18, 24, 30, 36, 42, 48, 54, 60, and 66 hours after dose (this schedule is q6h through Day 3, up to just prior to Day 4). In addition, sampling continues out through Day 70, on specific days, q12h.

Pharmacokinetics parameters: AUCs, Cmax, tmax, elimination half-life (t½), lag time (tlag), apparent clearance (CL/F) and apparent volume of distribution (V/F), area under the plasma drug concentration versus time curve on Days 1 through end of study (up to 70 Days)

Secondary Endpoints

pharmacodynamic effects of GSK2374697 in healthy subjects after meal challenge
On 2 days
dose proportionality of GSK2374697
up to 70 days post dose
Unlock Study Endpoints

Study Design & Arms

AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
GSK2376497ACTIVE_COMPARATORsingle dose escalation or multiple-dose titration
0.9% sodium chloridePLACEBO_COMPARATORplacebo injection

Interventions

NameTypeDescription
GSK2376497DRUGGSK2376497 Active Comparator
0.9% sodium chlorideDRUG0.9% sodium chloride Placebo Comparator
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy as determined by a responsible and experienced physician, based on a medical evaluation including medical history, physical examination, laboratory tests and Holter monitoring. A subject with a clinical abnormality or laboratory parameters outside the reference range f...

Countries:United States
Unlock Eligibility Criteria

Frequently asked questions about GSK2376497

What is GSK2376497 used for?

GSK2376497 is an investigational small molecule being developed for the treatment of Type 2 Diabetes Mellitus. It is currently in Phase 1 clinical development and has not been approved by regulatory authorities.

What does GSK2376497 target?

The molecular target of GSK2376497 has not been disclosed. It is being studied as a potential treatment for Type 2 Diabetes Mellitus, but its specific mechanism of action is not publicly available.

Who makes GSK2376497?

GSK2376497 is being developed by GSK plc, a global pharmaceutical company listed on the London Stock Exchange under the ticker GSK. The company is conducting clinical trials to evaluate the drug's safety and tolerability.

What phase is GSK2376497 in?

GSK2376497 is in Phase 1 clinical development. A Phase 1 study has been completed, and the drug remains investigational. It has not received regulatory approval and is still being evaluated for safety and tolerability.

What clinical trials is GSK2376497 in?

GSK2376497 has one completed Phase 1 clinical trial, NCT01545570, titled 'A Study to Determine the Safety, Tolerability, and Effects of GSK2374697 in Healthy Volunteers.' This trial enrolled 82 participants in the United States and was placebo-controlled, randomized, and double-blind.

Is GSK2376497 the same as GSK2374697?

The clinical trial NCT01545570 refers to GSK2374697, which appears to be a variant name for GSK2376497. The study evaluates the safety and tolerability of the compound in healthy volunteers for Type 2 Diabetes Mellitus.