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GSK2248761 WBM

Phase 1

Infections, Human Immunodeficiency Virus and Herpesviridae | Small molecule | Infectious Disease |GSK plc|Last Updated: Jun 8, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment24
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01209117A Study to Assess the Relative Bioavailability of Tablet Formulations of GSK2248761 in Healthy Adult Subjects. SGN114435PHASE1 COMPLETED 24Sep 1, 2010Jan 1, 2011Jun 8, 20171 United States
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Study Endpoints
Primary Endpoints
Plasma GSK2248761 Area under the concentration-time curve from time zero (pre-dose) extrapolated to infinite time (AUC(0-infinity))
5 weeks
Plasma GSK2248761 Area under the concentration-time curve over the dosing interval (AUC (0 - t))
5 weeks
Plasma GSK2248761 observed concentration 24 hours after dose (C24)
5 weeks
Plasma GSK2248761 Maximum observed concentration (Cmax)
5 weeks
Secondary Endpoints
Safety and tolerability parameters, including adverse events
5 weeks
concurrent medication
5 weeks
Clinical laboratory screens
5 weeks
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeOTHER
Treatment Arms
ArmTypeDescription
Periods 1 - 4EXPERIMENTALSubjects will be randomized in a cross over fashion to receive the GSK2248761 WBM capsule formulation or one of three WBM tablet formulations in one of four sequences.
Period 5EXPERIMENTALSubjects in Part B will receive a formulation of GSK2248761 200mg WBM Tablet chosen from Periods 1 - 4 in part A in the fed state (moderate fat meal).
Interventions
NameTypeDescription
GSK2248761 WBM CapsuleDRUG200 mg GSK2248761 WBM capsule (reference) 2 X100mg
GSK2248761 WBM Tablet Formulation 1DRUGGSK2248761 WBM Tablet 200mg manufacturing process 1
GSK2248761 WBM Tablet Formulation 2DRUGGSK2248761 WBM Tablet 200mg manufacturing process 2
GSK2248761 WBM Tablet Formulation 3DRUGGSK2248761 WBM Tablet 200mg manufacturing process 3
GSK2248761 WBM TabletDRUGGSK2248761 WBM tablet 200mg manufacturing process 1, 2, or 3 chosen from Period 1 - 4
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Eligibility Criteria
Age Range18 Years — 50 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy as determined by a responsible and experienced physician, based on a medical evaluation including medical history, physical examination, vital signs, laboratory tests, and ECGs. A subject with a clinical abnormality or laboratory parameters outside the reference range ...

Countries:United States
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