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GSK159802

Phase 1

Pulmonary Disease, Chronic Obstructive | Small molecule | Other |GSK plc|Last Updated: Sep 29, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment43
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00364273GSK159802 In Healthy Male Subjects And AsthmaticsPHASE1 COMPLETED 43Aug 24, 2005Jul 6, 2006Sep 29, 20172 United Kingdom
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Study Endpoints
Primary Endpoints
Safety & tolerability of single inhaled doses of GSK159802.
Up to 71 days
Secondary Endpoints
sGaw (Cohorts 1 and 2 only) and FEV1 Systemic & urine pharmacokinetics of GSK159802 and SKF-91300 Heart rate, potassium, glucose, 12-lead ECG & blood pressure
Up to 71 days
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Study Design & Arms
AllocationRANDOMIZED
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Subjects receiving treatment sequence 1 : Cohort 1EXPERIMENTALEligible subjects will receive placebo, GSK159802 300 micrograms, GSK159802 600 micrograms, GSK159802 900 micrograms and GSK159802 1200 micrograms.
Subjects receiving treatment sequence 2 : Cohort 1EXPERIMENTALEligible subjects will receive GSK159802 150 micrograms, placebo, GSK159802 600 micrograms, GSK159802 900 micrograms and GSK159802 1200 micrograms.
Subjects receiving treatment sequence 3 : Cohort 1EXPERIMENTALEligible subjects will receive GSK159802 150 micrograms, GSK159802 300 micrograms, placebo, GSK159802 900 micrograms and GSK159802 1200 micrograms.
Subjects receiving treatment sequence 4 : Cohort 1EXPERIMENTALEligible subjects will receive GSK159802 150 micrograms, GSK159802 300 micrograms, GSK159802 600 micrograms, placebo and GSK159802 1200 micrograms.
Subjects receiving treatment sequence 5 : Cohort 1EXPERIMENTALEligible subjects will receive GSK159802 150 micrograms, GSK159802 300 micrograms, GSK159802 600 micrograms, GSK159802 900 micrograms and placebo.
Subjects receiving treatment sequence 1 : Cohort 2EXPERIMENTALEligible subjects will receive placebo, salmeterol, GSK159802 low dose (LD) and GSK159802 maximum tolerated dose (MTD).
Subjects receiving treatment sequence 2 : Cohort 2EXPERIMENTALEligible subjects will receive salmeterol, GSK159802 MTD, placebo and GSK159802 LD.
Subjects receiving treatment sequence 3 : Cohort 2EXPERIMENTALEligible subjects will receive GSK159802 LD, placebo, GSK159802 MTD and salmeterol.
Subjects receiving treatment sequence 4 : Cohort 2EXPERIMENTALEligible subjects will receive GSK159802 MTD, GSK159802 LD, salmeterol and placebo.
Subjects receiving treatment sequence 1 : Cohort 3EXPERIMENTALEligible subjects will receive placebo, salmeterol, GSK159802 300 micrograms and GSK159802 1200 micrograms.
Subjects receiving treatment sequence 2 : Cohort 3EXPERIMENTALEligible subjects will receive salmeterol, GSK159802 1200 micrograms, placebo and GSK159802 300 micrograms.
Subjects receiving treatment sequence 3 : Cohort 3EXPERIMENTALEligible subjects will receive GSK159802 300 micrograms, placebo, GSK159802 1200 micrograms and salmeterol.
Subjects receiving treatment sequence 4 : Cohort 3EXPERIMENTALEligible subjects will receive GSK159802 1200 micrograms, GSK159802 300 micrograms, salmeterol and placebo.
Subjects receiving treatment sequence 5 : Cohort 3EXPERIMENTALEligible subjects will receive GSK159802 1200 micrograms, salmeterol, GSK159802 300 micrograms and placebo.
Interventions
NameTypeDescription
GSK159802DRUGGSK159802 will be available with dosing strengths of 75 microgram per blister and 300 microgram per blister administered using DISKUS inhaler.
PlaceboDRUGSubjects will receive placebo administered using DISKUS inhaler.
SalmeterolDRUGSalmeterol will be available with dosing strength of 50 micrograms per blister administered using DISKUS inhaler.
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Eligibility Criteria
Age Range18 Years — N/A
SexMALE
Healthy VolunteersYes
Study Sites2

Inclusion criteria: * Body mass index within the range 18.5-29.9 (kg/m2) * Current non-smokers who have not used any tobacco products in the 6-month period preceding the screening visit and have a pack history of \< 10 pack years. Additional criteria for Cohorts 2 and 3 only (Asthmatic Patients): ...

Countries:United Kingdom
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