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GSK1362885

Phase 1

Diabetes Mellitus, Type 2 | Small molecule | Metabolic |GSK plc|Last Updated: Jul 7, 2017

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials2
Total Enrollment65

FDA Designations

No designations recorded

Clinical trial landscape

GSK1362885 · 2 trials · 1 indication

Phase 1 2
NCT01013766A Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of GSK1362885 in Type 2 DiabeticsDiabetes Mellitus, Type 2
COMPLETED23 Analytics
NCT00823940A Phase 1 Study to Evaluate the Safety and Tolerability of GSK1362885 in Healthy Normal SubjectsDiabetes Mellitus, Type 2
COMPLETED42 Analytics
PHASE1COMPLETED
A Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of GSK1362885 in Type 2 Diabetics
Diabetes Mellitus, Type 2Unlock trial analytics
PHASE1COMPLETED
A Phase 1 Study to Evaluate the Safety and Tolerability of GSK1362885 in Healthy Normal Subjects
Diabetes Mellitus, Type 2Unlock trial analytics

Study Endpoints

Primary Endpoints

Safety and tolerability assessments including adverse events and clinical laboratory tests
7 Days
Pharmacodynamics following oral administration (glucose, insulin, c-peptide)
24 hours
Pharmacokinetic parameters: AUC, Cmax, Tmax, t1/2, tlag, Cl/F, and V/F
24 hours
Safety and tolerability assessments including adverse events, clinical laboratory tests, electrocardiogram (ECG) and vital signs
During the duration of study participation (from 2 days up to 5 weeks)

Secondary Endpoints

Pharmacodynamics following BID administration (glucose, insulin, c-peptide)
24 hours
Relationship between pharmacokinetic and pharmacodynamic parameters
24 hours
Pharmacokinetic parameters to assess dose proportionality and food effect
24 - 48 hours following each dose
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
AM/PM/BIDOTHERSubjects will receive a dose of 100mg in the AM on Day 1, followed by a dose of 100mg in the PM on Day 4, and a dose of 50mg BID on Day 6.
PM/AM/BIDOTHERSubjects will receive a dose of 100mg in the PM on Day 1, followed by a dose of 100mg in the AM on Day 4, followed by 50mg BID on Day 6.
Cohort A1PLACEBO_COMPARATORDose escalation: 5 - 100mg and placebo in 4 planned doses
Cohort A2PLACEBO_COMPARATORDose escalation: 100-600mg and placebo in 4 planned doses
Cohort B1OTHERGlucagon challenge test
Cohort B3ACTIVE_COMPARATORGlucagon challenge test + selected dose of GSK1362885

Interventions

NameTypeDescription
GSK1362885DRUG100mg in the AM, 100mg in the PM, 50mg BID
GlucagonDRUG0.5mg IV bolus
Glucagon + GSK1362885DRUG0.5mg Glucagon IV bolus + selected dose of GSK1362885
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersNo
Study Sites2

Inclusion Criteria: A subject will be eligible for inclusion in this study only if all of the following criteria apply: * A diagnosis of T2DM as determined by a responsible physician based on a medical evaluation including medical history, physical examination, and laboratory tests. Subjects may b...

Countries:United States
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Frequently asked questions about GSK1362885

What is GSK1362885 used for?

GSK1362885 is an investigational small molecule being developed for the treatment of Type 2 Diabetes Mellitus. It is in Phase 1 clinical development and is not yet approved by regulatory authorities. The drug is being studied for its safety, tolerability, pharmacokinetics, and pharmacodynamics in clinical trials.

Who makes GSK1362885?

GSK1362885 is being developed by GSK plc, a global biopharmaceutical company listed on the stock exchange under the ticker GSK. The company is conducting Phase 1 clinical trials to evaluate the drug's safety and tolerability in healthy subjects and in patients with Type 2 Diabetes Mellitus.

What phase is GSK1362885 in?

GSK1362885 is in Phase 1 clinical development. Two Phase 1 trials have been completed, involving a total of 65 participants. The drug is investigational and has not received regulatory approval. It is being studied for the treatment of Type 2 Diabetes Mellitus.

What clinical trials is GSK1362885 in?

GSK1362885 has been studied in two completed Phase 1 clinical trials. NCT00823940 evaluated safety and tolerability in healthy subjects with 42 participants. NCT01013766 evaluated safety, tolerability, pharmacokinetics, and pharmacodynamics in Type 2 diabetics with 23 participants. Both trials were conducted in the United States.

Is GSK1362885 FDA approved?

GSK1362885 is not FDA approved. It is an investigational drug currently in Phase 1 clinical development for Type 2 Diabetes Mellitus. The completed trials have evaluated its safety and tolerability, but the drug has not yet progressed through the later phases required for regulatory approval.