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GSK1362885

Phase 1

Diabetes Mellitus, Type 2 | Small molecule | Metabolic |GSK plc|Last Updated: Jul 7, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials2
Total Enrollment65
FDA Designations
No designations recorded
Clinical Trials (2)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01013766A Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of GSK1362885 in Type 2 DiabeticsPHASE1 COMPLETED 23Aug 13, 2009Nov 20, 2009Jun 20, 20172 United States
NCT00823940A Phase 1 Study to Evaluate the Safety and Tolerability of GSK1362885 in Healthy Normal SubjectsPHASE1 COMPLETED 42Jan 13, 2009Apr 27, 2009Jul 7, 20171 United States
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Study Endpoints
Primary Endpoints
Safety and tolerability assessments including adverse events and clinical laboratory tests
7 Days
Pharmacodynamics following oral administration (glucose, insulin, c-peptide)
24 hours
Pharmacokinetic parameters: AUC, Cmax, Tmax, t1/2, tlag, Cl/F, and V/F
24 hours
Safety and tolerability assessments including adverse events, clinical laboratory tests, electrocardiogram (ECG) and vital signs
During the duration of study participation (from 2 days up to 5 weeks)
Secondary Endpoints
Pharmacodynamics following BID administration (glucose, insulin, c-peptide)
24 hours
Relationship between pharmacokinetic and pharmacodynamic parameters
24 hours
Pharmacokinetic parameters to assess dose proportionality and food effect
24 - 48 hours following each dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
AM/PM/BIDOTHERSubjects will receive a dose of 100mg in the AM on Day 1, followed by a dose of 100mg in the PM on Day 4, and a dose of 50mg BID on Day 6.
PM/AM/BIDOTHERSubjects will receive a dose of 100mg in the PM on Day 1, followed by a dose of 100mg in the AM on Day 4, followed by 50mg BID on Day 6.
Cohort A1PLACEBO_COMPARATORDose escalation: 5 - 100mg and placebo in 4 planned doses
Cohort A2PLACEBO_COMPARATORDose escalation: 100-600mg and placebo in 4 planned doses
Cohort B1OTHERGlucagon challenge test
Cohort B3ACTIVE_COMPARATORGlucagon challenge test + selected dose of GSK1362885
Interventions
NameTypeDescription
GSK1362885DRUG100mg in the AM, 100mg in the PM, 50mg BID
GlucagonDRUG0.5mg IV bolus
Glucagon + GSK1362885DRUG0.5mg Glucagon IV bolus + selected dose of GSK1362885
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Eligibility Criteria
Age Range18 Years — 65 Years
SexALL
Healthy VolunteersNo
Study Sites2

Inclusion Criteria: A subject will be eligible for inclusion in this study only if all of the following criteria apply: * A diagnosis of T2DM as determined by a responsible physician based on a medical evaluation including medical history, physical examination, and laboratory tests. Subjects may b...

Countries:United States
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