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GSK1349572 formulation AP

Phase 1

Infection, Human Immunodeficiency Virus | Small molecule | Other |GSK plc|Last Updated: Jun 9, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLEDBiomarker
Total Trials1
Total Enrollment24
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01098513GSK1349572 Relative Bioavailability StudyPHASE1 COMPLETED 24Apr 1, 2010Jul 1, 2010Jun 9, 20171 United States
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Study Endpoints
Primary Endpoints
Plasma GSK1349572 AUC(0-infinity), AUC(0-t), and Cmax.
48 hours
Secondary Endpoints
Plasma GSK1349572 t½, tlag, tmax, C24, Vdss/F, CL/F, and MRT.
48 hours
Safety and tolerability parameters, including adverse events, concurrent medication, clinical laboratory screens, ECG, and vital signs assessments.
10 weeks
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part AEXPERIMENTALSubjects will be randomized in a three-way crossover design to receive a single dose of each of three different tablet formulations of GSK1349572 50 mg (2 tablets). Formulation AP, AW and AX.
Part BEXPERIMENTALA total of 18 subjects who complete Part A will return for Part B. Subjects from Part A will be asked to participate on a first come first served basis until there are 18 subjects, at which time enrolment to Part B will be closed. Part B will be a three way crossover design using either formulation AW or AX depending upon the results from Part A. Subjects will receive a single dose of 50 mg GSK1349572 with either a low fat, moderate fat or high fat meal in each period.
Interventions
NameTypeDescription
GSK1349572 formulation APDRUGGSK1349572 50 mg single dose fasted.
GSK1349572 formulation AWDRUGGSK1349572 formulation AW 50 mg single dose in Part A and 75 to 200 mg fasted or with moderate or high fat meal in Part B.
GSK1349572 formulation AXDRUGGSK1349572 formulation AX 50 mg in Part A and 75-200 mg fasted or with a moderate or high fat meal in Part B
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Eligibility Criteria
Age Range18 Years — 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * AST, ALT, alkaline phosphatase and bilirubin less than or equla to 1.5xULN (isolated bilirubin \>1.5xULN is acceptable if bilirubin is fractionated and direct bilirubin \<35%). * Healthy as determined by a responsible and experienced physician, based on a medical evaluation in...

Countries:United States
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