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GSBR-1290

Phase 1

Overweight or Obesity | Small molecule | Metabolic |Structure Therapeutics Inc.|Last Updated: Apr 25, 2024

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment142
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT05762471Phase 1b/2a Study of GSBR-1290 in Adult Overweight or Obese Healthy Subjects and Subjects With Type 2 Diabetes MellitusPHASE1 COMPLETED 142Jan 9, 2023Apr 11, 2024Apr 25, 20244 United States
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Study Endpoints
Primary Endpoints
Incidence, severity and relationship of AE/SAE, vital signs, laboratory measures and ECG to assess safety and tolerability of multiple oral doses of GSBR-1290 in HOV and T2DM
42 days
Secondary Endpoints
Analysis of Cmax at specified timepoints predose and postdose to calculate PK parameters
31 days
Analysis of Tmax at specified timepoints predose and postdose to calculate PK parameters
31 days
Analysis of AUC at specified timepoints predose and postdose to calculate PK parameters
31 days
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Cohort 1EXPERIMENTALPatients will receive once daily doses of study drug (GSBR-1290 or Placebo) for a total of 4 weeks
Cohort 2EXPERIMENTALPatients will receive once daily doses of study drug (GSBR-1290 or Placebo) for a total of 4 weeks
Cohort 3EXPERIMENTALPatients will receive once daily doses of study drug (GSBR-1290 or Placebo) for a total of 4 weeks
Cohort 4EXPERIMENTALHOV participants (Cohort 4) will receive multiple-ascending doses of GSBR-1290 or placebo for a total of 12 weeks
Cohort 5EXPERIMENTALParticipants with T2DM(Cohort 5) will be randomized to placebo, low-dose, or high-dose arms. Participants in the low-dose, high-dose or placebo arms will receive multiple-ascending doses for 12 weeks
Interventions
NameTypeDescription
GSBR-1290DRUGPatients will receive GSBR-1290 or matching Placebo
PlaceboDRUGPatients will receive GSBR-1290 or matching Placebo
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Eligibility Criteria
Age Range18 Years — 75 Years
SexALL
Healthy VolunteersNo
Study Sites4

Inclusion Criteria cohorts 1-4: 1. Provided evidence of a signed consent 2. Age ≥ 18 and ≤ 75 years 3. Healthy overweight/obese adult men and women with body mass index ≥ 27 and ≤ 40 kg/m2 4. No nicotine use 5. Have a suitable venous access for blood sampling Inclusion Criteria cohort 5: 1. Men a...

Countries:United States
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