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GEN1057

Phase 1

Advanced Malignant Solid Tumors | Small molecule | Oncology |Genmab A/S|Last Updated: Mar 2, 2026

Target and mechanism

Molecular targetDR4
Target classProtein
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment45

FDA Designations

No designations recorded

Clinical trial landscape

GEN1057 · 1 trial · 2 indications

Phase 1 1
NCT06573294Trial to Assess the Safety and Antitumor Activity of GEN1057 in Malignant Solid TumorsAdvanced Malignant Solid Tumors
RECRUITING45 Analytics
PHASE1RECRUITING
Trial to Assess the Safety and Antitumor Activity of GEN1057 in Malignant Solid Tumors
Advanced Malignant Solid TumorsUnlock trial analytics

Study Design & Arms

Interventions

NameTypeDescription
GEN1057DRUGIntravenous (IV) infusion
PremedicationDRUGIV infusion/orally by mouth.
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Frequently asked questions about GEN1057

What is GEN1057 used for?

GEN1057 is an investigational small molecule being developed for the treatment of advanced malignant solid tumors, including metastatic malignant solid tumors. It is currently in Phase 1 clinical development and has not been approved by regulatory authorities.

What does GEN1057 target?

GEN1057 targets DR4, a protein also known as death receptor 4. By targeting this protein, the drug is designed to potentially induce apoptosis, or programmed cell death, in tumor cells. This mechanism is being evaluated in the context of advanced solid tumors.

Who is developing GEN1057?

GEN1057 is being developed by Genmab A/S, a biotechnology company listed on the Nasdaq under the ticker symbol GMAB. The company is conducting clinical trials to assess the safety and antitumor activity of this investigational drug.

What phase is GEN1057 in?

GEN1057 is in Phase 1 clinical development. It is currently being studied in an early-stage trial to evaluate its safety, tolerability, and preliminary antitumor activity in patients with advanced malignant solid tumors. The drug is not yet approved for commercial use.

What clinical trials is GEN1057 in?

GEN1057 is being evaluated in a Phase 1 clinical trial with the identifier NCT06573294. This trial is titled 'Trial to Assess the Safety and Antitumor Activity of GEN1057 in Malignant Solid Tumors' and is currently recruiting participants with advanced or metastatic solid tumors.