Recent Updates
Recently added Catalysts

Tegobuvir

Phase 2

Hepatitis C, Chronic | Small molecule | Infectious Disease |Gilead Sciences, Inc.|Last Updated: Feb 6, 2014

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment245
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01271790A Study of Response-Guided Duration of Combination Therapy With GS-9451, Pegasys® and Copegus® With and Without Tegobuvir (GS-9190) in Previously Untreated Subjects With Genotype 1 Chronic Hepatitis CPHASE2 COMPLETED 245Oct 1, 2010Sep 1, 2013Feb 6, 2014144 United States, Austria +6
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Sustained virologic response
24 weeks of off-treatment follow-up

Sustained virologic response (SVR) defined as undetectable hepatitis C virus (HCV) RNA 24 weeks after treatment cessation

Secondary Endpoints
Safety and tolerability of therapy
Through treatment period and 24 weeks of off-treatment follow-up
Emergence of viral resistance following initiation of therapy with GS 9190 and GS 9451
Through treatment period, 24 weeks of off-treatment follow-up, and up to 48 weeks of follow-up in the Resistance Registry Substudy
Viral dynamics and steady state pharmacokinetics
Through Week 4 of therapy
Unlock Study Endpoints
Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Arm 1ACTIVE_COMPARATORGS-9451 and Tegobuvir (GS-9190) in combination with Pegasys® and Copegus® for 16 or 24 weeks; Pegasys® and Copegus® may be continued for up to 48 weeks total duration depending on individual response to therapy
Arm 2ACTIVE_COMPARATORGS-9451 (active) and Tegobuvir (GS-9190) placebo in combination with Pegasys® and Copegus® for 24 weeks; Pegasys® and Copegus® may be continued for up to 48 weeks total duration depending on individual response to therapy
Arm 3PLACEBO_COMPARATORPlacebo matching Tegobuvir (GS-9190) and GS-9451 in combination with Pegasys® and Copegus® for 24 weeks; Pegasys® and Copegus® will be continued for up to 48 weeks total duration
Interventions
NameTypeDescription
Tegobuvir (GS-9190)DRUGTegobuvir (GS-9190) capsule, 30 mg BID
GS-9451DRUGGS-9451 tablet, 200 mg once daily (QD)
Pegasys®BIOLOGICALpeginterferon alfa-2a (solution for injection) 180 µg/week
Copegus®DRUGribavirin tablet (weight based: 1000 mg/day \<75 kg; 1200 mg/day ≥ 75 kg) divided twice daily (BID)
Tegobuvir placeboDRUGplacebo matching Tegobuvir (GS-9190) capsule BID
GS-9451 placeboDRUGplacebo matching GS-9451 tablet QD
Unlock Study Design Details
Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersNo
Study Sites144

Inclusion Criteria: * Adult subjects 18 to 70 years of age * Chronic HCV infection for at least 6 months prior to Baseline (Day 1) * Liver biopsy results (performed no more than 2 years prior to Screening) indicating the absence of cirrhosis * Monoinfection with HCV genotype 1a or 1b * HCV treatmen...

Countries:United StatesAustriaBelgiumFranceGermanyNetherlandsPolandUnited Kingdom
Unlock Eligibility Criteria