Recent Updates
Recently added Catalysts

MBX-8025

Phase 2

Homozygous Familial Hypercholesterolemia | Small molecule | Metabolic |Gilead Sciences, Inc.|Last Updated: Mar 9, 2016

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
UNCONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment13
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT02472535Study to Evaluate the Effects of MBX-8025 in Patients With HoFHPHASE2 COMPLETED 13Apr 1, 2015Feb 1, 2016Mar 9, 20165 Canada, France +2
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
LDL-C
12-Weeks

Absolute and percentage (%) reduction in serum LDL-C at any point from baseline through Week 16.

Secondary Endpoints
Total Cholesterol (TC)
12-Weeks
High-density lipoprotein (HDL) cholesterol [HDL-C]
12-Weeks
Very Low-Density Lipoprotein (VLDL)
12-Weeks
Unlock Study Endpoints
Study Design & Arms
AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
placebo, MBX-8025 50 mg, 100 mg or 200 mg capsulesEXPERIMENTAL -
Interventions
NameTypeDescription
Run-In Period: PlaceboOTHER2 capsules, once a day for two weeks
MBX-8025 50 mg (Dose Escalation Period 1)DRUG1 capsule once a day for 4 weeks (MBX-8025 50 mg capsule)
MBX-8025 50 mg or 100 mg (Dose Escalation Period 2)DRUG1 capsule once a day for 4 weeks (MBX-8025 50 mg or 100 mg capsule)
MBX-8025 50 mg, 100 mg or 200 mg (Dose Escalation Period 3)DRUG1 or 2 capsules once a day for 4 weeks (MBX-8025 50 mg, 100 mg or two (2) 100 mg capsules)
Unlock Study Design Details
Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites5

Inclusion Criteria: 1. Must have given written informed consent (signed and dated) and any authorizations required by local law and be able to comply with all study requirements. 2. Male or female with HoFH confirmed by genotype (two mutant alleles at the LDL-Receptor (LDL-R) gene locus or double h...

Countries:CanadaFranceNetherlandsNorway
Unlock Eligibility Criteria