Recent Updates
Recently added Catalysts

belapectin

Phase 1

Hepatic Impairment | Small molecule | Gastrointestinal |Galectin Therapeutics Inc.|Last Updated: Mar 28, 2022

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
UNCONTROLLEDBiomarker
Total Trials1
Total Enrollment38
FDA Designations
FAST_TRACK
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04332432A Single-dose, Open-label, Pharmacokinetic Study of Belapectin (GR-MD-02) in Subjects With Normal Hepatic Function and Subjects With Varying Degrees of Hepatic ImpairmentPHASE1 COMPLETED 38Jun 16, 2020Mar 9, 2022Mar 28, 20224 United States
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Area under the concentration-time curve from time 0 to infinity (AUC0-∞) (Blood)
Blood samples for pharmacokinetics will be taken on Day -1, and on Day 1 at pre dose, 2, 3, 4, 24, 36, 48, 72, 96, 120, 216 (Day 10), and 336 (Day 15) hours post dose (post-end of infusion).
Area under the concentration-time curve from time 0 to infinity (AUC0-∞) (Urine)
Urine samples for pharmacokinetics will be taken on Day -1 (spot sample), at pre-dose (spot sample) on Day 1 and at the following intervals: 2 to 4, 4 to 24, 24 to 36, 36 to 48, 48 to 72, 72 to 96, and 96 to 120 hours post-dose.
Area under the concentration-time curve from time 0 to the last measurable concentration (AUC0-t) (Blood)
Blood samples for pharmacokinetics will be taken on Day -1, and on Day 1 at pre dose, 2, 3, 4, 24, 36, 48, 72, 96, 120, 216 (Day 10), and 336 (Day 15) hours post dose (post-end of infusion).
Area under the concentration-time curve from time 0 to the last measurable concentration (AUC0-t) (Urine)
Urine samples for pharmacokinetics will be taken on Day -1 (spot sample), at pre-dose (spot sample) on Day 1 and at the following intervals: 2 to 4, 4 to 24, 24 to 36, 36 to 48, 48 to 72, 72 to 96, and 96 to 120 hours post-dose.
Maximum observed concentration (Cmax) (Blood)
Blood samples for pharmacokinetics will be taken on Day -1, and on Day 1 at pre dose, 2, 3, 4, 24, 36, 48, 72, 96, 120, 216 (Day 10), and 336 (Day 15) hours post dose (post-end of infusion).
Maximum observed concentration (Cmax) (Urine)
Urine samples for pharmacokinetics will be taken on Day -1 (spot sample), at pre-dose (spot sample) on Day 1 and at the following intervals: 2 to 4, 4 to 24, 24 to 36, 36 to 48, 48 to 72, 72 to 96, and 96 to 120 hours post-dose.
Time of the maximum observed concentration (tmax) (Blood)
Blood samples for pharmacokinetics will be taken on Day -1, and on Day 1 at pre dose, 2, 3, 4, 24, 36, 48, 72, 96, 120, 216 (Day 10), and 336 (Day 15) hours post dose (post-end of infusion).
Time of the maximum observed concentration (tmax) (Urine)
Urine samples for pharmacokinetics will be taken on Day -1 (spot sample), at pre-dose (spot sample) on Day 1 and at the following intervals: 2 to 4, 4 to 24, 24 to 36, 36 to 48, 48 to 72, 72 to 96, and 96 to 120 hours post-dose.
Terminal elimination half-life (t½) (Blood)
Blood samples for pharmacokinetics will be taken on Day -1, and on Day 1 at pre dose, 2, 3, 4, 24, 36, 48, 72, 96, 120, 216 (Day 10), and 336 (Day 15) hours post dose (post-end of infusion).
Terminal elimination half-life (t½) (Urine)
Urine samples for pharmacokinetics will be taken on Day -1 (spot sample), at pre-dose (spot sample) on Day 1 and at the following intervals: 2 to 4, 4 to 24, 24 to 36, 36 to 48, 48 to 72, 72 to 96, and 96 to 120 hours post-dose.
Time of last measurable concentration (tlast) (Blood)
Blood samples for pharmacokinetics will be taken on Day -1, and on Day 1 at pre dose, 2, 3, 4, 24, 36, 48, 72, 96, 120, 216 (Day 10), and 336 (Day 15) hours post dose (post-end of infusion).
Time of last measurable concentration (tlast) (Urine)
Urine samples for pharmacokinetics will be taken on Day -1 (spot sample), at pre-dose (spot sample) on Day 1 and at the following intervals: 2 to 4, 4 to 24, 24 to 36, 36 to 48, 48 to 72, 72 to 96, and 96 to 120 hours post-dose.
Total clearance (CL) (Blood)
Blood samples for pharmacokinetics will be taken on Day -1, and on Day 1 at pre dose, 2, 3, 4, 24, 36, 48, 72, 96, 120, 216 (Day 10), and 336 (Day 15) hours post dose (post-end of infusion).
Total clearance (CL) (Urine)
Urine samples for pharmacokinetics will be taken on Day -1 (spot sample), at pre-dose (spot sample) on Day 1 and at the following intervals: 2 to 4, 4 to 24, 24 to 36, 36 to 48, 48 to 72, 72 to 96, and 96 to 120 hours post-dose.
Apparent volume of distribution at steady state (Vss) (Blood)
Blood samples for pharmacokinetics will be taken on Day -1, and on Day 1 at pre dose, 2, 3, 4, 24, 36, 48, 72, 96, 120, 216 (Day 10), and 336 (Day 15) hours post dose (post-end of infusion).
Apparent volume of distribution at steady state (Vss) (Urine)
Urine samples for pharmacokinetics will be taken on Day -1 (spot sample), at pre-dose (spot sample) on Day 1 and at the following intervals: 2 to 4, 4 to 24, 24 to 36, 36 to 48, 48 to 72, 72 to 96, and 96 to 120 hours post-dose.
Secondary Endpoints
Incidence and severity of AEs
Screening through end of study (Day 15)
Incidence of laboratory abnormalities
Screening through end of study (Day 15)
Unlock Study Endpoints
Study Design & Arms
AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
belapectinEXPERIMENTALSingle dose of 4 mg/kg of lean body mass (LBM) belapectin solution for injection administered intravenously (infused over approximately 60 minutes). Group 1: 16 matched healthy subjects with normal hepatic function Group 2: 8 subjects with mild hepatic impairment (Child-Pugh Class A \[4 x subjects with a score of 5 and 4 x subjects with a score of 6\]) Group 3: 8 subjects with moderate hepatic impairment (Child-Pugh Class B \[score of 7 to 9\]) Group 4: 8 subjects with severe hepatic impairment (Child-Pugh Class C \[score of 10 to 14\]).
Interventions
NameTypeDescription
belapectinDRUGintravenous
Unlock Study Design Details
Eligibility Criteria
Age Range18 Years — 75 Years
SexALL
Healthy VolunteersYes
Study Sites4

Inclusion Criteria: All Subjects 1. Males or females, of any race, between 18 and 75 years of age, inclusive. 2. Body mass index between 18.0 and 45.0 kg/m2, inclusive. 3. Females of childbearing potential will not be pregnant or lactating and must have a negative result on an approved pregnancy t...

Countries:United States
Unlock Eligibility Criteria