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Nafamostat Mesilate

Phase 1

Pharmacokinetics | Small molecule | Other |Ensysce Biosciences, Inc.|Last Updated: Sep 24, 2024

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment17
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04406415Oral Nafamostat in Healthy Volunteers (NAF-101)PHASE1 COMPLETED 17Sep 21, 2020May 14, 2021Sep 24, 20241 United States
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Study Endpoints
Primary Endpoints
Safety and Tolerability
14 Days

Number of participants with adverse events including out-of-range clinical laboratory measures, vital signs, ECG, and spontaneous adverse event reports throughout the 14 day study period

Secondary Endpoints
Pharmacokinetics (Cmax)
Pre-dose (0 hr) and at 0.5, 1, 2, 3, 4, 6, and 8 hr after first dose on Day 1 and again after the last dose on Day 5
Pharmacokinetics (Tmax)
Pre-dose (0 hr) and at 0.5, 1, 2, 3, 4, 6, and 8 hr after first dose on Day 1 and again after the last dose on Day 5
Pharmacokinetics (AUC)
Pre-dose (0 hr) and at 0.5, 1, 2, 3, 4, 6, and 8 hr after first dose on Day 1 and again after the last dose on Day 5
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Study Design & Arms
AllocationRANDOMIZED
MaskingSINGLE
ModelSEQUENTIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
10 mgEXPERIMENTAL10 mg nafamostat three times a day (t.i.d., approximately q8h) for up to 5 days
50 mgEXPERIMENTAL50 mg nafamostat three times a day (t.i.d., approximately q8h) for up to 5 days
100 mgEXPERIMENTAL100 mg nafamostat three times a day (t.i.d., approximately q8h) for up to 5 days
200 mgEXPERIMENTAL200 mg nafamostat three times a day (t.i.d., approximately q8h) for up to 5 days
PlaceboPLACEBO_COMPARATORPlacebo administered three times a day (t.i.d., approximately q8h) for up to 5 days
Interventions
NameTypeDescription
Nafamostat MesilateDRUGOral nafamostat, 10, 50, 100, or 200 mg administered three times daily for up to 5 days
PlaceboDRUGOral placebo administered three times daily for up to 5 days
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Eligibility Criteria
Age Range18 Years — 70 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Males or females, age 18 to 70 years old, able and willing to provide written informed consent to participate in the study; 2. Subjects must be in generally good health as determined by pre-study medical history, physical examination, clinical laboratory tests, and 12-lead el...

Countries:United States
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