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VLX-1005

Phase 1

Heparin-induced Thrombocytopenia | Small molecule | Hematology |Cadrenal Therapeutics, Inc.|Last Updated: Jan 11, 2023

Success Probability

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Market & Valuation

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Trial Design

RandomizedACTIVE_CONTROLLEDBiomarker
Total Trials1
Total Enrollment12

FDA Designations

ORPHAN_DRUGFAST_TRACK

Clinical trial landscape

VLX-1005 · 2 trials · 2 indications

Phase 1 2
NCT05325346A Phase I Study of the Co-administration of VLX-1005 and Argatroban in Healthy Human SubjectsHeparin-induced Thrombocytopenia
COMPLETED12 Analytics
NCT04783545Phase I Study of VLX-1005 in Healthy SubjectsSafety and Tolerability in Healthy Volunteers
COMPLETED96 Analytics
PHASE1COMPLETED
A Phase I Study of the Co-administration of VLX-1005 and Argatroban in Healthy Human Subjects
Heparin-induced ThrombocytopeniaUnlock trial analytics
PHASE1COMPLETED
Phase I Study of VLX-1005 in Healthy Subjects
Safety and Tolerability in Healthy VolunteersUnlock trial analytics

Study Endpoints

Primary Endpoints

Effects of argatroban on Cmax of VLX-1005
0 - 51 hours

Measure the effects of argatroban on the maximum plasma concentration (Cmax) of VLX-1005

Effects of VLX-1005 on Cmax of argatroban
0 - 51 hours

Measure the effects of VLX-1005 on the maximum plasma concentration (Cmax) of argatroban

Effects of argatroban on Tmax of VLX-1005
0 - 51 hours

Measure the effects of argatroban on the time to maximum plasma concentration (Tmax) of VLX-1005

Effects of VLX-1005 on Tmax of argatroban
0 - 51 hours

Measure the effects of VLX-1005 on the time to maximum plasma concentration (Tmax) of argatroban

Effects of argatroban on AUC(inf) of VLX-1005
0 - 51 hours

Measure the effects of argatroban on the Area Under the Curve \[AUC(inf)\] of VLX-1005

Effects of VLX-1005 on AUC(inf) of argatroban
0 - 51 hours

Measure the effects of VLX-1005 on the Area Under the Curve \[AUC(inf)\] of argatroban

Effects of VLX-1005 on whole blood aggregometry
0 - 9 hours

The change in impedance from baseline by whole blood aggregometry will be measured to assess the effects of VLX-1005 on platelet aggregation

Effects of argatroban on whole blood aggregometry
0 - 9 hours

The change in impedance from baseline by whole blood aggregometry will be measured to assess the effects of argatroban on platelet aggregation

Effects of VLX-1005 on PFA-100
0 - 9 hours

Change in PFA-100 (a platelet pharmacodynamic measure) from baseline, to assess the effects of VLX-1005 on platelet aggregation

Effects of argatroban on PFA-100
0 - 9 hours

Change in PFA-100 (a platelet pharmacodynamic measure) from baseline, to assess the effects of argatroban on platelet aggregation

Number of Participants Reporting One or More Treatment-emergent Adverse Events
Baseline up to Day 29
Number of Participants Who Meet the Markedly Abnormal Criteria for Vital Sign Measurements at Least Once Post Dose
Baseline up to Day 29
Number of Participants Who Meet the Markedly Abnormal Criteria for 12-lead Electrocardiogram (ECG) or Telemetry Parameters at Least Once Post Dose
Baseline up to Day 29
Number of Participants Who Meet the Markedly Abnormal Criteria for Laboratory Values at Least Once Post Dose
Baseline up to Day 29

Secondary Endpoints

Safety as measured by incidence of Treatment Emergent Adverse Events
0 - 30 days
Effects of VLX-1005 on 12-HETE
0 - 12 hours
Effects of argatroban on 12-HETE
0 - 12 hours
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
VLX-1005EXPERIMENTALIntravenous administration of VLX-1005 with measurements of PK and PD
ArgatrobanACTIVE_COMPARATORIntravenous administration of argatroban with measurements of PK and PD
VLX-1005 and ArgatrobanOTHERIntravenous co-administration of VLX-1005 and argatroban with measurements of PK and PD
Single Ascending Dose Cohorts 1-6EXPERIMENTALDrug: VLX-1005
Single Ascending Dose Cohorts 1-6, PlaceboPLACEBO_COMPARATORDrug: Placebo
Multiple Ascending Dose Cohorts 7-9EXPERIMENTALDrug: VLX-1005
Multiple Ascending Dose Cohorts 7-9, PlaceboPLACEBO_COMPARATORDrug: Placebo

Interventions

NameTypeDescription
VLX-1005DRUGMeasurement and comparison of the effects and potential interactions between VLX-1005 and argatroban on safety, tolerability, PK and PD
ArgatrobanDRUGMeasurement and comparison of the effects and potential interactions between VLX-1005 and argatroban on safety, tolerability, PK and PD
PlaceboDRUGPlacebo infusion
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Eligibility Criteria

Age Range19 Years to 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Healthy, adult, male or female (non-lactating and not of childbearing potential) subjects age 19 to 55 inclusive. 2. Females must have undergone one of the following sterilization procedures at least 6 months prior to the first dosing: 1. hysteroscopic sterilization 2....

Countries:United States
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Frequently asked questions about VLX-1005

What is VLX-1005 used for?

VLX-1005 is an investigational small molecule being developed for heparin-induced thrombocytopenia, a condition related to blood clotting. It is also being studied for safety and tolerability in healthy volunteers. The drug is in Phase 1 clinical development and has not been approved by the FDA.

What does VLX-1005 target?

VLX-1005 is a small molecule being developed by Cadrenal Therapeutics for heparin-induced thrombocytopenia. The specific molecular target of VLX-1005 has not been disclosed in available information. The drug is currently in Phase 1 clinical trials to evaluate its safety and tolerability.

Who makes VLX-1005?

Cadrenal Therapeutics, Inc. (NASDAQ: CVKD) is developing VLX-1005. The company is conducting Phase 1 clinical trials for this investigational small molecule, which is being studied for heparin-induced thrombocytopenia and safety in healthy volunteers.

What phase is VLX-1005 in?

VLX-1005 is in Phase 1 clinical development. It has completed two Phase 1 trials, including one studying its co-administration with argatroban in healthy subjects. The drug is investigational and has not received FDA approval. It has been granted orphan drug and fast track designations.

What clinical trials is VLX-1005 in?

VLX-1005 has completed two Phase 1 trials. NCT04783545 studied VLX-1005 in 96 healthy subjects in the United States. NCT05325346 studied co-administration of VLX-1005 and argatroban in 12 healthy subjects for heparin-induced thrombocytopenia. Both trials are completed.

Is VLX-1005 the same as argatroban?

No, VLX-1005 is not the same as argatroban. VLX-1005 is an investigational small molecule being developed by Cadrenal Therapeutics. Argatroban is a separate anticoagulant medication. A Phase 1 trial (NCT05325346) studied the co-administration of both drugs in healthy subjects.