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CORT125281

Phase 1

Healthy | Small molecule | Other |Corcept Therapeutics Incorporated|Last Updated: Jul 26, 2018

Target and mechanism

ModalitySmall molecule

Also known as CORT125281, 40mg, fasted, CORT125281, fasted

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment48

FDA Designations

No designations recorded

Clinical trial landscape

CORT125281 · 1 trial · 1 indication

Phase 1 1
NCT03335956CORT125281 Single Ascending Dose (SAD) and Multiple Ascending Dose (MAD)Healthy
COMPLETED48 Analytics
PHASE1COMPLETED
CORT125281 Single Ascending Dose (SAD) and Multiple Ascending Dose (MAD)
HealthyUnlock trial analytics

Study Endpoints

Primary Endpoints

Adverse Events (AEs)
SAD Cohorts Day 1 to Day 14; MAD Cohorts Day 1 to Day 30

Secondary Endpoints

AUCtau Pharmacokinetic (PK) parameter
MAD Cohorts Day 3 to 19
AUC 0-tz PK parameter
CORT125281/CORT125324 - SAD Cohorts Day 1 to 4; MAD Cohorts Day 3 to 19; Pioglitizone - MAD Cohort Day 1 to 15
AUC 0-infinity PK parameter
CORT125281/CORT125324 - SAD Cohorts Day 1 to 4; MAD Cohorts Day 3 to 19; Pioglitizone - MAD Cohort Day 1 to 15
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Study Design & Arms

AllocationRANDOMIZED
MaskingTRIPLE
ModelPARALLEL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
SAD Part 1 Placebo Cohort 1 Period 1PLACEBO_COMPARATOR -
SAD Part 1 Active Cohort Period 1EXPERIMENTAL -
SAD Part 1 Placebo Cohort 1 Period 2PLACEBO_COMPARATOR -
SAD Part 1 Active Cohort 1 Period 2EXPERIMENTAL -
SAD Part 1 Placebo Cohort 1 Period 3PLACEBO_COMPARATOR -
SAD Part 1 Active Cohort 1 Period 3EXPERIMENTAL -
SAD Part 2 Placebo Cohort 2 Period 4PLACEBO_COMPARATOR -
SAD Part 2 Active Cohort 2 Period 4EXPERIMENTAL -
SAD Part 2 Placebo Cohort 2 Period 5PLACEBO_COMPARATOR -
SAD Part 2 Active Cohort 2 Period 5EXPERIMENTAL -
SAD Part 2 Placebo Cohort 2 Period 6PLACEBO_COMPARATOR -
SAD Part 2 Active Cohort 2 Period 6EXPERIMENTAL -
MAD Placebo Cohort 1PLACEBO_COMPARATOR -
MAD Active Cohort 1EXPERIMENTAL -
MAD Placebo Cohort 2PLACEBO_COMPARATOR -
MAD Active Cohort 2EXPERIMENTAL -
MAD Placebo Cohort 3PLACEBO_COMPARATOR -
MAD Active Cohort 3EXPERIMENTAL -
MAD Placebo Cohort 4PLACEBO_COMPARATOR -
MAD Active Cohort 4EXPERIMENTAL -

Interventions

NameTypeDescription
CORT125281, 40mg, fastedDRUGCORT125281 is supplied as capsules for oral dosing
Prednisone 25mg, fastedDRUGChallenge Agent, Dose and Route of Administration: Standard release 25 mg tablets, orally administered
Placebo oral capsule, fastedDRUGReference Therapy, Dose and Route of Administration: Placebo capsule, orally administered
Pioglitazone 15mg TabletDRUGProbe Substrate, Dose and Route of Administration: 15 Mg tablet, orally administered
Placebo oral capsule, fedDRUGReference Therapy, Dose and Route of Administration: Placebo capsule, orally administered
Prednisone 25mg, fedDRUGChallenge Agent, Dose and Route of Administration: Standard release 25 mg tablets, orally administered
CORT125281, 120mg, fastedDRUGCORT125281 is supplied as capsules for oral dosing
CORT125281, 360mg, fastedDRUGCORT125281 is supplied as capsules for oral dosing
CORT125281, 720mg, fastedDRUGCORT125281 is supplied as capsules for oral dosing
CORT125281, 360mg, fedDRUGCORT125281 is supplied as capsules for oral dosing
CORT125281, 360mgDRUGCORT125281 is supplied as capsules for oral dosing twice, 12 hours apart, fasted (morning) and after evening meal
CORT125281, 120mgDRUGCORT125281 is supplied as capsules for oral dosing once daily
CORT125281, 180mgDRUGCORT125281 is supplied as capsules for oral dosing twice daily
CORT125281, 240mgDRUGCORT125281 is supplied as capsules for oral dosing twice daily
Placebo oral capsuleDRUGReference Therapy, Dose and Route of Administration: Placebo capsule, orally administered twice, 12 hours apart, fasted (morning) and after evening meal
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: 1. Give written informed consent 2. If male, have undergone vasectomy, with no wish to have the procedure reversed 3. If female, using appropriate precautions to avoid pregnancy, defined as of nonchildbearing potential (ie, postmenopausal or permanently sterilised) or using high...

Countries:United Kingdom
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Frequently asked questions about CORT125281

What is CORT125281 used for?

CORT125281 is an investigational small molecule being studied in healthy volunteers. It is currently in Phase 1 clinical development, with a completed trial evaluating single and multiple ascending doses. The drug is being developed by Corcept Therapeutics Incorporated.

What does CORT125281 target?

CORT125281 is a small molecule developed by Corcept Therapeutics. The specific molecular target has not been disclosed in available clinical trial information. The drug is being studied in healthy volunteers to assess its safety, tolerability, and pharmacokinetics.

Who makes CORT125281?

CORT125281 is being developed by Corcept Therapeutics Incorporated, a biopharmaceutical company. The company is conducting clinical trials to evaluate the drug's safety and tolerability in healthy volunteers.

What phase is CORT125281 in?

CORT125281 is in Phase 1 clinical development. A Phase 1 trial studying single ascending doses (SAD) and multiple ascending doses (MAD) has been completed. The drug is investigational and has not been approved by regulatory authorities.

What clinical trials is CORT125281 in?

CORT125281 has one completed Phase 1 clinical trial, identified as NCT03335956, titled "CORT125281 Single Ascending Dose (SAD) and Multiple Ascending Dose (MAD)." The trial enrolled 48 healthy volunteers in the United Kingdom and was randomized, double-blind, and placebo-controlled.