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Rasigiline

Phase 1

Healthy Volunteers | Small molecule | Other |Bristol-Myers Squibb Company|Last Updated: Aug 31, 2023

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment128
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04978298Study to Evaluate the Pressor Effect of Oral Tyramine During Ozanimod Treatment in Healthy Adult ParticipantsPHASE1 COMPLETED 128Jul 19, 2021Feb 26, 2023Aug 31, 20231 United States
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Study Endpoints
Primary Endpoints
Tyramine Sensitivity Factor (TSF)
Up to Day 85

The ratio of Tyramine pressor response (Tyr30) in Period 1 over Tyr30 in Period 3.

Secondary Endpoints
Heart Rate (HR)
Up to Day 85
Systolic Blood Pressure (SBP)
Up to Day 85
Diastolic Blood Pressure (DBP)
Up to Day 85
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Rasagiline groupEXPERIMENTALParticipants will receive rasagiline once daily (QD) for 14 days from Days 59 to 72.
Phenelzine groupEXPERIMENTALParticipants will receive phenelzine twice daily (BID) for 14 days from Days 59 to 72.
Ozanimod Therapeutic groupEXPERIMENTALParticipants will receive ozanimod QD for 65 days (including the initial 7-day dose escalation) from Days 8 to 72.
Ozanimod Supra-therapeutic groupEXPERIMENTALParticipants will receive ozanimod QD for 65 days (including the initial 10-day dose escalation) from Days 8 to 72.
PlaceboPLACEBO_COMPARATORParticipants will receive matched appropriate placebos from Days 8 to 72.
Interventions
NameTypeDescription
PlaceboOTHERPlacebo
RasigilineDRUGRasigiline
PhenelzineDRUGPhenelzine
OzanimodDRUGOzanimod
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Eligibility Criteria
Age Range25 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: Participants must satisfy the following criteria to be enrolled in the study: 1. Be a male or non-pregnant, non-lactating female, 25 to 55 years of age, inclusive, at the time of signing the informed consent form. 2. Must understand and voluntarily sign an informed consent form...

Countries:United States
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