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Nintedanib

Phase 1

Healthy Participants | Small molecule | Other |Bristol-Myers Squibb Company|Last Updated: Mar 14, 2025

Target and mechanism

Molecular targetPDGFRB, PDGFRA, FLT1, FLT4, KDR, FGFR3, FGFR1, FGFR4, FGFR2
Target classInhibitor
ModalitySmall molecule

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment71

FDA Designations

No designations recorded

Clinical trial landscape

Nintedanib · 1 trial · 1 indication

Phase 1 1
NCT06568458A Study to Assess the Extent of Drug Interaction Between BMS-986278 and Nintedanib, the Relative Bioavailability of BMS-986278 in Tablet and the Effect That Food Has on BMS-986278 in Tablet Formulations in Healthy ParticipantsHealthy Participants
COMPLETED71 Analytics
PHASE1COMPLETED
A Study to Assess the Extent of Drug Interaction Between BMS-986278 and Nintedanib, the Relative Bioavailability of BMS-986278 in Tablet and the Effect That Food Has on BMS-986278 in Tablet Formulations in Healthy Participants
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Study Endpoints

Primary Endpoints

Maximum Observed Serum Concentration (Cmax)
Days 4, 17, 21 (Part-1); Days 1, 7, 13 (Part-2); Days 1, 7 (Part-3)
Area under the plasma concentration-time curve within a dosing interval AUC(TAU)
Day 4, 17 and 21 of Part 1
Area under the plasma concentration-time curve from time zero to time of last quantifiable concentration AUC(0-T)
Day 1-6 (part-2 and Part-3), Day 7-12 (Part2 and 3), Day 13-18) (Part-2)
Area under the plasma concentration-time curve from time zero extrapolated to infinite time AUC(INF)
Day 1-6 (part-2 and Part-3), Day 7-12 (Part2 and 3), Day 13-18) (Part-2)

Secondary Endpoints

Number of participants with non-serious AEs (Adverse events)
Up to 28 Days post discontinuation of dosing
Number of participants with Serious AEs
Up to 28 Days post discontinuation of dosing
Number of participants with AEs leading to discontinuation
Up to 28 Days post discontinuation of dosing
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Part I: Period AEXPERIMENTAL -
Part I: Period BEXPERIMENTAL -
Part I: Period CEXPERIMENTAL -
Part II: Period 1EXPERIMENTAL -
Part II: Period 2EXPERIMENTAL -
Part II: Period 3EXPERIMENTAL -
Part III: Period 1EXPERIMENTAL -
Part III: Period 2EXPERIMENTAL -

Interventions

NameTypeDescription
NintedanibDRUGSpecified Dose on specified days
BMS 986278DRUGSpecified dose on specified days
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Eligibility Criteria

Age Range18 Years to 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Participants must be healthy males and females (INOCBP) * Participant must have Body mass index (BMI) of 18.0 kg/m2 through 32.0 kg/m2, inclusive. * Participant must have Body weight ≥ 50 kg Exclusion Criteria: * Participant must not have current or recent GI disease * Parti...

Countries:United States
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Frequently asked questions about Nintedanib

What is Nintedanib used for in Healthy Participants?

Nintedanib is a small molecule being studied in healthy participants to assess drug interactions and bioavailability. A completed Phase 1 trial evaluated the extent of drug interaction between BMS-986278 and Nintedanib, the relative bioavailability of BMS-986278 in tablet form, and the effect of food on tablet formulations. It is investigational and not approved for this use.

What does Nintedanib target?

Nintedanib targets multiple receptor tyrosine kinases, including PDGFRB, PDGFRA, FLT1, FLT4, KDR, FGFR3, FGFR1, FGFR4, and FGFR2. It acts as an inhibitor of these targets, which are involved in signaling pathways related to cell growth and angiogenesis.

Who makes Nintedanib?

Nintedanib is being developed by Bristol-Myers Squibb Company, traded under the ticker BMY. The company is conducting clinical research on the drug, including a Phase 1 trial in healthy participants.

What phase is Nintedanib in?

Nintedanib is in Phase 1 clinical development. The single trial listed is a completed Phase 1 study with 71 participants. It is an investigational drug and has not been approved for any indication based on the available data.

What clinical trials is Nintedanib in?

Nintedanib has one completed clinical trial, NCT06568458, a Phase 1 study in healthy participants in the United States. The trial assessed drug interactions between BMS-986278 and Nintedanib, the relative bioavailability of BMS-986278 tablets, and the effect of food on tablet formulations. Enrollment was 71 participants.