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BMS-986259

Phase 2

Acute Decompensated Heart Failure | Small molecule | Cardiovascular |Bristol-Myers Squibb Company|Last Updated: Aug 4, 2022

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment25

FDA Designations

No designations recorded

Clinical trial landscape

BMS-986259 · 3 trials · 3 indications

Phase 2 1Phase 1 2
NCT04318093Study of the Safety of BMS-986259 in Participants With Post-Acute Decompensated Heart FailureAcute Decompensated Heart Failure
COMPLETED25 Analytics
PHASE2COMPLETED
Study of the Safety of BMS-986259 in Participants With Post-Acute Decompensated Heart Failure
Acute Decompensated Heart FailureUnlock trial analytics

Study Endpoints

Primary Endpoints

Percentage of Participants Experiencing Clinically Relevant Hypotension
From first dose to 30 days following first dose

Clinically Relevant Hypotension is defined as occurrence of any of the following: * Supine Systolic Blood Pressure (SBP) \<85 mmHg (confirmed by repeat measurement within 30 minutes), regardless of symptoms of hypotension * Supine SBP \<90 mmHg (confirmed by repeat measurement within 30 minutes) AND symptoms of hypotension (eg, dizziness, lightheadedness, etc).

Maximum plasma Concentration (Cmax) of BMS-986259 in Blood serum
Day 1 and Day 8
Time to reach maximum concentration in plasma (Tmax) of BMS-986259 in blood serum
Day 1 and Day 8
Area under the concentration- time curve over the dosing interval of BMS-986259 in blood serum - AUC(TAU)
Day 1 and Day 8
Concentration of BMS-986259 in blood serum at 24 hours (C24)
Day 1 and Day 8
Area under the concentration-time curve of BMS-986259 from time 0 (dosing) to the time of the last quantifiable - AUC(0-T)
Day 8
Accumulation ratio in the maximum plasma concentration of BMS-986259 in blood serum -AR(Cmax)
Day 8
Accumulation ratio of Area under the concentration-time curve in BMS-986259 over the dosing interval -AR (AUC [TAU])
Day 8
Accumulation ratio concentration of BMS-986259 at 24 hours- AR(C24)
Day 8
Terminal elimination half-life of BMS-986259 (T-HALF)
Day 8
Apparent total clearance of BMS-986259 at steady-state (CLss/F)
Day 8
Apparent volume of distribution of BMS-986259 at terminal phase at steady-state (Vss/F)
Day 8
Incidence of Adverse Events (AEs)
Up to 7 weeks
Incidence of Serious Adverse Events (SAEs)
up to 7 weeks
AEs leading to discontinuation
Up to 7 weeks
Number of clinically significant changes in vital signs
Up to 7 weeks
Number of clinically significant changes in ECG (electrocardiogram)
Up to 7 weeks
Number of clinically significant changes in physical examinations
Up to 7 weeks
Number of clinically significant changes in clinical laboratory tests
Up to 7 weeks

Secondary Endpoints

Maximum Observed Serum Concentration (Cmax)
Day 1 and Day 5 of study treatment
Time of Maximum Observed Serum Concentration (Tmax)
Day 1 and Day 5 of study treatment
Area Under the Concentration-Time Curve Within a Dosing Interval (AUC(TAU))
Day 1 and Day 5 of study treatment
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Study Design & Arms

AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
BMS-986259EXPERIMENTAL -
PlaceboPLACEBO_COMPARATOR -
Arm A: Normal Renal FunctionEXPERIMENTAL -
Arm B: Mild Renal ImpairmentEXPERIMENTAL -
Arm C: Moderate Renal ImpairmentEXPERIMENTAL -
Arm D: Severe Renal ImpairmentEXPERIMENTAL -
Part A SAD - A1 CohortEXPERIMENTALSingle Ascending Dose
Part A SAD - A2 CohortEXPERIMENTALSingle Ascending dose
Part A SAD- A3 CohortEXPERIMENTALSingle Ascending dose
Part A SAD- A4 CohortEXPERIMENTALSingle Ascending dose
Part A SAD - A5 CohortEXPERIMENTALSingle Ascending dose
Part A SAD- A6 CohortEXPERIMENTALSingle Ascending dose
Part B MAD- B1 CohortEXPERIMENTALMultiple Ascending Dose
Part B MAD - B2 CohortEXPERIMENTALMultiple Ascending Dose
Part B MAD - B3 CohortEXPERIMENTALMultiple Ascending Dose
Part B MAD - B4 CohortEXPERIMENTALMultiple Ascending Dose
Part C JMAD - C1 CohortEXPERIMENTALJapanese Multiple Ascending Dose
Part C JMAD - C2 CohortEXPERIMENTALJapanese Multiple Ascending Dose
Part C JMAD - C3 CohortEXPERIMENTALJapanese Multiple Ascending Dose

Interventions

NameTypeDescription
BMS-986259DRUGSpecified dose on specified days
PlaceboOTHERSpecified dose on specified days
P-AminohippurateDIAGNOSTIC_TESTDiagnostic Agent
IohexolDIAGNOSTIC_TESTDiagnostic Agent
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites18

For more information regarding Bristol-Myers Squibb Clinical Trial participation, please visit www.BMSStudyConnect.com Inclusion Criteria: * Participants currently hospitalized for acute decompensated heart failure (ADHF) * Participants must be hemodynamically stable, as assessed by the investigat...

Countries:ArgentinaCzechiaGreeceIsraelPolandUnited KingdomUnited StatesNetherlands
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Frequently asked questions about BMS-986259

What is BMS-986259 used for?

BMS-986259 is an investigational small molecule being studied for acute decompensated heart failure, renal failure, and in healthy participants. It is in clinical development by Bristol-Myers Squibb. The drug has completed Phase 1 and Phase 2 trials, but it is not approved and remains under investigation.

Who makes BMS-986259?

BMS-986259 is being developed by Bristol-Myers Squibb Company, which trades under the ticker BMY. The company has sponsored clinical trials of the drug in healthy participants, in participants with renal failure, and in participants with post-acute decompensated heart failure.

What phase is BMS-986259 in?

BMS-986259 is in Phase 2 clinical development. A Phase 2 study of the drug in participants with post-acute decompensated heart failure has been completed. Earlier Phase 1 trials in healthy participants and in participants with renal failure have also been completed. The drug is investigational and not yet approved.

What clinical trials has BMS-986259 been in?

BMS-986259 has been studied in three completed clinical trials. NCT04008992 was a Phase 1 ascending dose study in healthy participants. NCT04237831 was a Phase 1 study in participants with various levels of kidney function. NCT04318093 was a Phase 2 study in participants with post-acute decompensated heart failure.

Is BMS-986259 FDA approved?

BMS-986259 is not FDA approved. It is an investigational drug that has completed Phase 1 and Phase 2 clinical trials. The drug is still in clinical development for acute decompensated heart failure and related conditions, and its safety and efficacy have not been established for regulatory approval.