Recent Updates
Recently added Catalysts

Pecavaptan

Phase 1

Congestive Heart Failure | Small molecule | Cardiovascular |Bayer AG|Last Updated: Oct 31, 2022

Success Probability

Subscribe to view

Market & Valuation

Subscribe to view

Trial Design

CONTROLLED
Total Trials1
Total Enrollment32

FDA Designations

No designations recorded

Clinical trial landscape

Pecavaptan · 1 trial · 2 indications

Phase 1 1
NCT05599997A Study to Learn How the Study Treatment BAY1753011 Moves Into, Through and Out of the Body, How it Works, How Safe it is, and How it Affects the Body When Given Once as Tablet in Male and Female Participants With Reduced Kidney Function Compared to Matched Participants With Normal Kidney FunctionCongestive Heart Failure
COMPLETED32 Analytics
PHASE1COMPLETED
A Study to Learn How the Study Treatment BAY1753011 Moves Into, Through and Out of the Body, How it Works, How Safe it is, and How it Affects the Body When Given Once as Tablet in Male and Female Participants With Reduced Kidney Function Compared to Matched Participants With Normal Kidney Function
Congestive Heart FailureUnlock trial analytics

Study Endpoints

Primary Endpoints

Area under the concentration versus time curve from zero to infinity divided by dose of total BAY1753011 in plasma after single dose administration (AUC/D)
From pre-dose until 144 hours post dose

Dose-normalized AUC (AUC/D) of BAY1753011 was investigated as the dose for the severe renal impairment group was reduced to 15 mg.

Maximum observed drug concentration divided by dose of total BAY1753011 in plasma after single dose administration (Cmax/D)
From pre-dose until 144 hours post dose

Dose-normalized Cmax (Cmax/D) of BAY1753011 was investigated as the dose for the severe renal impairment group was reduced to 15 mg.

Area under the concentration versus time curve from zero to infinity divided by dose of unbound BAY1753011 in plasma after single dose administration (AUCu/D)
From pre-dose until 144 hours post dose

Dose-normalized AUCu (AUCu/D) of BAY1753011 was investigated as the dose for the severe renal impairment group was reduced to 15 mg.

Maximum observed drug concentration divided by dose of unbound BAY1753011 in plasma after single dose administration (Cmax,u/D)
From pre-dose until 144 hours post dose

Dose-normalized Cmax,u (Cmax,u/D) of BAY1753011 was investigated as the dose for the severe renal impairment group was reduced to 15 mg.

Secondary Endpoints

Number of participants with treatment-emergent adverse events
After first application of study medication up to 10 days after the study medication
Unlock Study Endpoints

Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
HealthyEXPERIMENTALAge-, weight- and gender- matched control group of healthy volunteers received a single oral dose of 30 mg BAY1753011 tablet.
Mild renal impairmentEXPERIMENTALSubjects with mild renal impairment received a single oral dose of 30 mg BAY1753011 tablet.
Moderate renal impairmentEXPERIMENTALSubjects with moderate renal impairment received a single oral dose of 30 mg BAY1753011 tablet.
Severe renal impairmentEXPERIMENTALSubjects with severe renal impairment received a single oral dose of 15 mg BAY1753011 tablet.

Interventions

NameTypeDescription
Pecavaptan (BAY1753011)DRUG30 mg, immediate release tablet, single dose, oral
Unlock Study Design Details

Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: * Male or female White participants (women without childbearing potential) * Aged from ≥18 years * body mass index above or equal 18.5 kg/m2 and below or equal 36 kg/m2 at the first screening visit * Participants with renal impairment: with an eGFR \<90 mL/min/1.73 m\^2 determin...

Countries:Germany
Unlock Eligibility Criteria

Frequently asked questions about Pecavaptan

What is Pecavaptan used for?

Pecavaptan is an investigational small molecule being developed for congestive heart failure. It is currently in Phase 1 clinical development and has not been approved by the FDA. The drug is being studied in patients with reduced kidney function, as well as in healthy volunteers.

Who makes Pecavaptan?

Pecavaptan is being developed by Bayer AG, a German pharmaceutical company. Bayer's stock is traded under the ticker symbol BAYRY on the OTC market. The drug is currently in Phase 1 clinical development for congestive heart failure.

What phase is Pecavaptan in?

Pecavaptan is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 study has been completed, which evaluated the drug's safety, tolerability, and pharmacokinetics in participants with reduced kidney function compared to those with normal kidney function.

What clinical trials is Pecavaptan in?

Pecavaptan has one completed Phase 1 clinical trial registered as NCT05599997. This study, conducted in Germany, enrolled 32 participants and evaluated how the drug moves into, through, and out of the body, as well as its safety and effects, in participants with reduced kidney function compared to matched participants with normal kidney function.

Is Pecavaptan the same as BAY1753011?

Yes, Pecavaptan is also known as BAY1753011. The Phase 1 clinical trial NCT05599997 refers to the study treatment as BAY1753011. This alternative name is used in the clinical trial registration and may appear in scientific literature and regulatory documents.