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BAY1237592

Phase 1

Hypertension, Pulmonary | Small molecule | Cardiovascular |Bayer AG|Last Updated: May 7, 2025

Success Probability

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Market & Valuation

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Trial Design

CONTROLLED
Total Trials1
Total Enrollment38

FDA Designations

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Clinical trial landscape

BAY1237592 · 1 trial · 1 indication

Phase 1 1
NCT03754660This Study Tests the Safety of Inhaled BAY1237592, How the Drug is Tolerated and How it Effects Patients With High Blood Pressure in the Arteries of the Lungs in the Two Different Disease Groups Pulmonary Arterial Hypertension (PAH) and Chronic Thromboembolic Pulmonary Hypertension (CTEPH)Hypertension, Pulmonary
COMPLETED38 Analytics
PHASE1COMPLETED
This Study Tests the Safety of Inhaled BAY1237592, How the Drug is Tolerated and How it Effects Patients With High Blood Pressure in the Arteries of the Lungs in the Two Different Disease Groups Pulmonary Arterial Hypertension (PAH) and Chronic Thromboembolic Pulmonary Hypertension (CTEPH)
Hypertension, PulmonaryUnlock trial analytics

Study Endpoints

Primary Endpoints

Peak percent reduction in PVR (Pulmonary vascular resistance) from "baseline 2" for untreated patients
Up to 5 hours post inhalation of BAY1237592 compared to "baseline 2"

PVR = 80\* (PAP - PCWP) / CO (dyn·sec·cm-5) * PAP = pulmonary arterial pressure * PCWP = pulmonary capillary wedge pressure * CO = cardiac output

Peak percent reduction in PVR from "baseline" for pre-treated patients
Up to 5 hours post inhalation of BAY1237592 compared to "baseline"

PVR = 80\* (PAP - PCWP) / CO (dyn·sec·cm-5)

Secondary Endpoints

Incidence of treatment-emergent adverse events (TEAEs)
Up to 7 days after treatment
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Study Design & Arms

AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
Untreated patients (Part A and Part B)EXPERIMENTALPart A: Untreated PAH and CTEPH patients will be enrolled to test 5 ascending doses of BAY1237592 with 4 patients per dose group up to a maximum dose of 4000 µg. Part B: The highest safe, well tolerated and effective dose of Part A will be tested in further untreated patients.
Monotherapy (Part B)EXPERIMENTALThe highest safe, well tolerated and effective dose chosen from Part A will be tested in pre-treated patients with any kind of monotherapy for PAH/CTEPH.
Combined therapy (Part B)EXPERIMENTALThe highest safe, well tolerated and effective dose from Part A will be tested in pre-treated patients with any kind of double combination treatment for PAH/CTEPH.

Interventions

NameTypeDescription
BAY1237592DRUGOral inhalation with dry powder inhaler, single dose.
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Eligibility Criteria

Age Range18 Years to 80 Years
SexALL
Healthy VolunteersNo
Study Sites8

Main Inclusion Criteria: * Patients with PAH or CTEPH undergoing medically indicated routine invasive diagnostics * Men and women aged 18 to 80 years Part A: \- Untreated patients: Therapy-naïve patients (defined as off treatment with PDE-5 inhibitors, endothelin receptor antagonists, prostanoids...

Countries:AustriaCzechiaGermanyPoland
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Frequently asked questions about BAY1237592

What is BAY1237592 used for?

BAY1237592 is an investigational small molecule being developed for pulmonary hypertension, specifically for two disease groups: pulmonary arterial hypertension (PAH) and chronic thromboembolic pulmonary hypertension (CTEPH). It is administered by inhalation and is currently in Phase 1 clinical development.

Who is developing BAY1237592?

BAY1237592 is being developed by Bayer AG, a German pharmaceutical company traded on the OTC market under the ticker BAYRY. The drug is in Phase 1 clinical development for pulmonary hypertension.

What phase is BAY1237592 in?

BAY1237592 is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 trial has been completed, and the drug is not currently in active clinical trials.

What clinical trials is BAY1237592 in?

BAY1237592 has one completed Phase 1 clinical trial, identified as NCT03754660. This study tested the safety, tolerability, and effects of inhaled BAY1237592 in patients with pulmonary arterial hypertension (PAH) and chronic thromboembolic pulmonary hypertension (CTEPH). The trial enrolled 38 participants across Austria, Czechia, Germany, and Poland.

How is BAY1237592 administered?

BAY1237592 is administered by inhalation. The completed Phase 1 trial (NCT03754660) tested the safety and tolerability of the inhaled formulation in patients with pulmonary arterial hypertension (PAH) and chronic thromboembolic pulmonary hypertension (CTEPH).