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BAY1002670_Vilaprisan

Phase 1

Endometriosis | Small molecule | Endocrine |Bayer AG|Last Updated: Jul 2, 2017

Success Probability

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Trial Design

UNCONTROLLED
Total Trials1
Total Enrollment12

FDA Designations

No designations recorded

Clinical trial landscape

BAY1002670_Vilaprisan · 1 trial · 1 indication

Phase 1 1
NCT02975440Drug-drug Interaction Study Between Orally Administered Rifampicin and VilaprisanEndometriosis
COMPLETED12 Analytics
PHASE1COMPLETED
Drug-drug Interaction Study Between Orally Administered Rifampicin and Vilaprisan
EndometriosisUnlock trial analytics

Study Endpoints

Primary Endpoints

AUC of Vilaprisan in plasma with co-medication Rifampicin
blood sampling for pharmacokinetics of Vilaprisan (LC-MS/MS) at the following time points post administration of Vilaprisan and Midazolam: 0.5,1,1.5,2,2.5,3,3.5,4,4.5,5,6,8,12,15 hour, thereafter daily sampling up to 14 days
Cmax of Vilaprisan in plasma with co-medication Rifampicin
blood sampling for pharmacokinetics of Vilaprisan (LC-MS/MS) at the following time points post administration of Vilaprisan and Midazolam: 0.5,1,1.5,2,2.5,3,3.5,4,4.5,5,6,8,12,15 hour, thereafter daily sampling up to 14 days
AUC of Vilaprisan in plasma without co-medication Rifampicin
blood sampling for pharmacokinetics of Vilaprisan (LC-MS/MS) at the following time points post administration of Vilaprisan and Midazolam: 0.5,1,1.5,2,2.5,3,3.5,4,4.5,5,6,8,12,15 hour, thereafter daily sampling up to 14 days
Cmax of Vilaprisan in plasma without co-medication Rifampicin
blood sampling for pharmacokinetics of Vilaprisan (LC-MS/MS) at the following time points post administration of Vilaprisan and Midazolam: 0.5,1,1.5,2,2.5,3,3.5,4,4.5,5,6,8,12,15 hour, thereafter daily sampling up to 14 days
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeBASIC_SCIENCE

Treatment Arms

ArmTypeDescription
TreatmentEXPERIMENTALTreatment A (Period 1): a single oral dose of 4 mg Vilaprisan and 1 mg Midazolam Treatment B (Period 2): 600 mg Rifampicin once daily (qd) for 7 days followed by administration of a single oral dose of 4 mg Vilaprisan and 1 mg Midazolam followed by 600 mg Rifampicin 12 hours after Vilaprisan and Midazolam administration and continued dosing of 600 mg Rifampicin once daily for 3 days

Interventions

NameTypeDescription
RifampicinDRUG11 single oral doses of 600 mg Rifampicin resulting in a total dose of 6600 mg Rifampicin.
MidazolamDRUG2 single oral doses of 1 mg Midazolam resulting in a total dose of 2 mg Midazolam
BAY1002670_VilaprisanDRUG2 single oral doses of 4 mg Vilaprisan resulting in a total dose of 8 mg Vilaprisan
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Eligibility Criteria

Age Range45 Years to 65 Years
SexFEMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy female postmenopausal subjects * Age: 45 to 65 years (inclusive) * Body mass index (BMI) : ≥20 and ≤32 kg/m² * Race: White Exclusion Criteria: * Any finding of the medical examination (including blood pressure, pulse rate and ECG) deviating from normal and of clinica...

Countries:Germany
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