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BAY 86-7660, levomefolate calcium

Phase 1

Pharmacology, Clinical | Small molecule | Other |Bayer AG|Last Updated: Aug 1, 2016

Success Probability

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Market & Valuation

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Trial Design

RandomizedACTIVE_CONTROLLED
Total Trials1
Total Enrollment43

FDA Designations

No designations recorded

Clinical trial landscape

BAY 86-7660, levomefolate calcium · 1 trial · 1 indication

Phase 1 1
NCT00941057Bioequivalence Study: 2 mg Estradiol Valerate (EV) and 3 mg Dienogest (DNG) Without and With Levomefolate CalciumPharmacology, Clinical
COMPLETED43 Analytics
PHASE1COMPLETED
Bioequivalence Study: 2 mg Estradiol Valerate (EV) and 3 mg Dienogest (DNG) Without and With Levomefolate Calcium
Pharmacology, ClinicalUnlock trial analytics

Study Endpoints

Primary Endpoints

AUC
Pre-dose and up to 72 hr post-dose for the treatments A and B and up to 12 hr post dose for the treatment C

Area under the concentration vs time curve from zero to infinity for DNG

Cmax
Pre-dose and up to 72 hr post-dose for the treatments A and B and up to 12 hr post dose for the treatment C

Maximum drug concentration for DNG and for E1, E2, E1S, and L-5-methyl-THF (baseline corrected and uncorrected)

AUC(0-tlast)
Pre-dose and up to 72 hr post-dose for the treatments A and B and up to 12 hr post dose for the treatment C

AUC from time 0 to the last data point above the lower limit of quantitation for E1, E2, E1S, and L-5-methyl-THF (baseline corrected and uncorrected)

Secondary Endpoints

tmax
Pre-dose and up to 72 hr post-dose for the treatments A and B and up to 12 hr post dose for the treatment C
Pre-dose and up to 72 hr post-dose for the treatments A and B and up to 12 hr post dose for the treatment C
λz
Pre-dose and up to 72 hr post-dose for the treatments A and B and up to 12 hr post dose for the treatment C
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Study Design & Arms

AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER

Treatment Arms

ArmTypeDescription
Estradiol + dienogest + levomefolateEXPERIMENTALTreatment A
Estradiol + dienogestACTIVE_COMPARATORTreatment B
LevomefolateACTIVE_COMPARATORTreatment C

Interventions

NameTypeDescription
BAY 98-7079, Estradiolvalerate (EV) / Dienogest (DNG) / Levomefolate calciumDRUGOral, single dose, 2 mg EV + 3 mg DNG + 0.451 mg levomefolate calcium washout phase between treatments: at least 7 days
BAY 86-5027,Estradiolvalerate(EV) / Dienogest (DNG)DRUGOral, single dose, 2 mg EV + 3 mg DNG washout phase between treatments: at least 7 days
BAY 86-7660,levomefolate calciumDRUGOral, single dose, 0.451 mg levomefolate calcium washout phase between treatments: at least 7 days
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Eligibility Criteria

Age Range45 Years to 75 Years
SexFEMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy postmenopausal women, age: 45-75 years with body mass index between ≥18 and ≤30 kg/m2. Post-menopausal state revealed by: medical history, and hormone analyses in serum: estradiol ≤20 pg/mL and in women \<60 years old: follicle-stimulating hormone ≥ 40 IU/L at screenin...

Countries:Germany
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Frequently asked questions about BAY 86-7660, levomefolate calcium

What is BAY 86-7660 used for?

BAY 86-7660, also known as levomefolate calcium, is a small molecule being investigated for pharmacology and clinical applications. It is currently in Phase 1 clinical development. The drug has been studied in a bioequivalence trial involving healthy female volunteers aged 45 years and older.

Who makes BAY 86-7660?

BAY 86-7660 is being developed by Bayer AG, a German pharmaceutical company. Bayer's stock is traded over-the-counter under the ticker symbol BAYRY. The drug is currently in Phase 1 clinical development.

What phase is BAY 86-7660 in?

BAY 86-7660 is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities. One Phase 1 clinical trial has been completed, and the drug is not currently in any active trials.

What clinical trials is BAY 86-7660 in?

BAY 86-7660 has been studied in one completed Phase 1 clinical trial, identified as NCT00941057. This was a bioequivalence study comparing 2 mg estradiol valerate and 3 mg dienogest with and without levomefolate calcium. The trial enrolled 43 healthy female volunteers in Germany.

Is BAY 86-7660 the same as levomefolate calcium?

Yes, BAY 86-7660 is also known as levomefolate calcium. The drug is being developed by Bayer AG and is currently in Phase 1 clinical development for pharmacology and clinical applications.