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ABI-H3733 Liquid Dosage Form

Phase 1

Chronic Hepatitis B | Small molecule | Infectious Disease |Assembly Biosciences, Inc.|Last Updated: Jan 27, 2021

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment120
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04271592A Study to Assess Safety, Tolerability, and Pharmacokinetics of ABI-H3733 in Healthy AdultsPHASE1 COMPLETED 120May 17, 2020Jan 14, 2021Jan 27, 20211 New Zealand
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Study Endpoints
Primary Endpoints
Number of Participants with One or More Adverse Events
Up to Day 10
Number of Participants with One or More Related Adverse Events
Up to Day 10
Number of Participants with One or More Severe (Grade ≥3) Adverse Events
Up to Day 10
Secondary Endpoints
SAD Cohorts 1-7: Area Under the Plasma Concentration Time Curve (AUC) of ABI-H3733
before and at pre-specified time points up to 120 hours after dosing
SAD Cohorts 1-7: Maximum Plasma Concentration (Cmax) ABI-H3733
before and at pre-specified time points up to 120 hours after dosing
SAD Cohorts 1-7: Time of Cmax (Tmax) of ABI-H3733
before and at pre-specified time points up to 120 hours after dosing
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelSEQUENTIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part 1: SAD Cohorts 1-7 ABI-H3733 Liquid FormEXPERIMENTALA single dose of ABI-H3733 liquid oral dosage form administered on Day 1. Cohort 1 will receive a 100-mg dose. Subsequent cohorts 2-7 will receive a ≤3-fold increase in dose from the previous cohort; the dose will be determined by evaluation of safety and PK data from previous cohorts.
Part 1: SAD Cohorts 1-7 Placebo Liquid FormPLACEBO_COMPARATORA single dose of placebo matching ABI-H3733 liquid oral dosage form will be administered on Day 1. Cohort 1 will receive a 100-mg dose. Subsequent cohorts 2-7 will receive a ≤3-fold increase in dose from the previous cohort; the dose will be determined by evaluation of safety and PK data from previous cohorts.
Part 1: MAD Cohorts 8-10 ABI-H3733 Liquid FormEXPERIMENTALOnce-daily doses of ABI-H3733 liquid oral dosage form will be administered from Day 1 to Day 5. Cohort 8 will receive a dose determined from evaluation of the data from the SAD cohorts. Subsequent cohorts 9 and 10 will receive a ≤3-fold increase in dose from the previous cohort; the dose will be determined by evaluation of safety and PK data from previous cohorts.
Part 1: MAD Cohorts 8-10 Placebo Liquid FormPLACEBO_COMPARATOROnce-daily doses of placebo matching ABI-H3733 liquid oral dosage form will be administered from Day 1 to Day 5. Cohort 8 will receive a dose determined from evaluation of the data from the SAD cohorts. Subsequent cohorts 9 and 10 will receive a ≤3-fold increase in dose from the previous cohort; the dose will be determined by evaluation of safety and PK data from previous cohorts.
Part 2: Single Dose Fasted Cohort 11 ABI-H3733 Solid FormEXPERIMENTALA single dose of ABI-H3733 solid oral dosage form will be administered in a fasted state on Day 1. The decision to proceed with Part 2 and the dose administered will be determined after evaluation of cumulative safety and PK data from Part 1.
Part 2: Single Dose Fasted Cohort 11 Placebo Solid FormPLACEBO_COMPARATORA single dose of placebo matching ABI-H3733 liquid oral dosage form will be administered in a fasted state on Day 1. The decision to proceed with Part 2 and the dose administered will be determined after evaluation of cumulative safety and PK data from Part 1.
Part 2: Single Dose Fed Cohort 12 ABI-H3733 Solid FormEXPERIMENTALA single dose of ABI-H3733 solid oral dosage form will be administered after a high-fat meal on Day 1. The decision to proceed with Part 2 and the dose administered will be determined after evaluation of cumulative safety and PK data from Part 1.
Part 2: Single Dose Fed Cohort 12 Placebo Solid FormPLACEBO_COMPARATORA single dose of placebo matching ABI-H3733 solid oral dosage form will be administered after a high-fat meal on Day 1. The decision to proceed with Part 2 and the dose administered will be determined after evaluation of cumulative safety and PK data from Part 1.
Interventions
NameTypeDescription
ABI-H3733 Liquid Oral Dosage FormDRUGABI-H3733 liquid oral dosage form
ABI-H3733 Solid Oral Dosage FormDRUGABI-H3733 solid oral dosage form
Placebo to ABI-H3733 Liquid Oral Dosage FormDRUGPlacebo to ABI-H3733 liquid oral dosage form
Placebo to ABI-H3733 Solid Oral Dosage FormDRUGPlacebo to ABI-H3733 solid oral dosage form
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Eligibility Criteria
Age Range18 Years — 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * No clinically significant abnormal findings on physical exam, medical history, or clinical laboratory results at screening. Exclusion Criteria: * Positive test results for human immunodeficiency virus (HIV) or hepatitis B or C. * History of or current persistent drug or alco...

Countries:New Zealand
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