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ALS-4

Phase 1

Healthy Subject | Small molecule | Other |Aptorum Group Limited|Last Updated: Apr 25, 2022

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment72
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT05274802A Study of ALS-4 in Healthy Adults SubjectsPHASE1 COMPLETED 72Mar 20, 2021Jan 2, 2022Apr 25, 20221 Canada
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Study Endpoints
Primary Endpoints
Number of participants with Adverse Events
Up to 28 days

An adverse event is any unfavorable and unintended sign (including a clinically significant abnormal laboratory finding, for example), symptom, or disease temporally associated with the Study or use of investigational drug product, whether or not the AE is considered related to the investigational drug product.

Secondary Endpoints
Area under the plasma concentration-time curve from time-zero extrapolated to infinite time (AUCinf)
Up to 24 hours post dose
Area under the plasma concentration vs time curve from time 0 to the time of the last measurable concentration, or last sampling time t (AUCt)
Up to 24 hours post dose
Time of maximum observed plasma concentration (Cmax)
Up to 24 hours post dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingTRIPLE
ModelSEQUENTIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part A1 (Single dose): Cohort A: ALS-4 25mgEXPERIMENTALSingle dose of ALS-4 or placebo before Breakfast
Part A1 (Single dose): Cohort B: ALS-4 50mgEXPERIMENTALSingle dose of ALS-4 or placebo before Breakfast
Part A1 (Single dose): Cohort C: ALS-4 100mgEXPERIMENTALSingle dose of ALS-4 or placebo before Breakfast
Part A1 (Single dose): Cohort D: ALS-4 200mgEXPERIMENTALSingle dose of ALS-4 or placebo before Breakfast
Part A1 (Single dose): Cohort E: ALS-4 300mgEXPERIMENTALSingle dose of ALS-4 or placebo before Breakfast
Part A2 (Single dose): Cohort F: ALS-4 50mgEXPERIMENTALDose three separate times in crossover fashion: (1) fasted morning dose; (2) fed morning dose; (3) fasted evening dose
Part B (Multiple dose): Cohort AA: ALS-4 50mgEXPERIMENTALMultiple dose of ALS-4 or placebo up to two times daily
Part B (Multiple dose): Cohort BB: ALS-4 100mgEXPERIMENTALMultiple dose of ALS-4 or placebo up to two times daily
Part B (Multiple dose): Cohort CC: ALS-4 200mgEXPERIMENTALMultiple dose of ALS-4 or placebo up to two times daily
Interventions
NameTypeDescription
ALS-4DRUGSingle dose of ALS-4 before Breakfast
PlaceboDRUGSingle dose of placebo before Breakfast
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Eligibility Criteria
Age Range18 Years — 60 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy, non-smoking male and female volunteers (18-60 years inclusive at the time of informed consent.) * Body mass index (BMI) within 18.5 - 33.0 kg/m2 inclusive and weight \>50 kg. * Healthy, according to the medical history, ECG, vital signs, laboratory results and physica...

Countries:Canada
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