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Olopatadine, 0.7%

Phase 3

Allergic Conjunctivitis | Small molecule | Ophthalmology |Alcon Inc.|Last Updated: Nov 17, 2017

Target and mechanism

ModalitySmall molecule

Also known as Olopatadine hydrochloride ophthalmic solution, 0.7%, Olopatadine Hydrochloride Nasal Spray 0.6%, Olopatadine 0.6%, Olopatadine Hydrochloride Ophthalmic Solution, 0.2%, Olopatadine, 0.2%, Olopatadine hydrochloride ophthalmic solution, 0.2%, Olopatadine 0.6% nasal spray, Olopatadine Hydrochloride Ophthalmic Solution 0.2%

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials5
Total Enrollment1,097

FDA Designations

No designations recorded

Clinical trial landscape

Olopatadine, 0.7% · 8 trials · 4 indications

Phase 3 6Phase 2 1Phase 1 1
NCT02322216Olopatadine Hydrochloride Ophthalmic Solution Study in Chinese SubjectsAllergic Conjunctivitis
COMPLETED383 Analytics
NCT01037179An Open-Label, Long-Term Study With AL-4943A Ophthalmic Solution, 0.2% in Patients With Allergic ConjunctivitisAllergic Conjunctivitis
COMPLETED110 Analytics
NCT00987272Study of Olopatadine HCl Ophthalmic Solutions Compared to Vehicle Using the Conjunctival Allergen Challenge (CAC) Model of Acute Allergic Conjunctivitis in Japanese SubjectsAllergic Conjunctivitis
COMPLETED267 Analytics
NCT00578929Safety and Efficacy of Olopatadine HCl Nasal Spray in 6-11 Year Old PatientsSeasonal Allergic Rhinitis
COMPLETED2,388 Analytics
NCT00578331Safety Study of Olopatadine Nasal SprayPerennial Allergic Rhinitis
COMPLETED890 Analytics
NCT00331500Olopatadine 0.2% for the Treatment of Allergic ConjunctivitisAllergic Conjunctivitis
COMPLETED287 Analytics
PHASE3COMPLETED
Olopatadine Hydrochloride Ophthalmic Solution Study in Chinese Subjects
Allergic ConjunctivitisUnlock trial analytics
PHASE3COMPLETED
An Open-Label, Long-Term Study With AL-4943A Ophthalmic Solution, 0.2% in Patients With Allergic Conjunctivitis
Allergic ConjunctivitisUnlock trial analytics
PHASE3COMPLETED
Study of Olopatadine HCl Ophthalmic Solutions Compared to Vehicle Using the Conjunctival Allergen Challenge (CAC) Model of Acute Allergic Conjunctivitis in Japanese Subjects
Allergic ConjunctivitisUnlock trial analytics
PHASE3COMPLETED
Safety and Efficacy of Olopatadine HCl Nasal Spray in 6-11 Year Old Patients
Seasonal Allergic RhinitisUnlock trial analytics
PHASE3COMPLETED
Safety Study of Olopatadine Nasal Spray
Perennial Allergic RhinitisUnlock trial analytics
PHASE3COMPLETED
Olopatadine 0.2% for the Treatment of Allergic Conjunctivitis
Allergic ConjunctivitisUnlock trial analytics

Study Endpoints

Primary Endpoints

Change From Baseline in Worst Ocular Itching Score During the 24 Hours Prior at Day 14
Baseline, Day 14

Severity of ocular itching was evaluated as the worst score observed in the past 24 hours prior to each study visit. Ocular itching was assessed by the participant on a scale from 0-4, where 0=None and 4=Incapacitating itch. One eye (study eye) contributed to the analysis.

Mean Itching Score by Visit
Up to Week 10

Ocular itching will be assessed by the subject and graded on a 6-point scale, where 0=did not occur and 5=virtually all the time over the past 3 days.

Mean Total Hyperemia Score by Visit
Up to Week 10

Ocular hyperemia (redness) will be assessed by the investigator. Total hyperemia score is defined as the sum of the palpebral and bulbar conjunctival scores.

Mean Ocular Itching Score
Day 0 of treatment: 3, 5, and 10 minutes post CAC
Percent Change From Baseline in the Reflective Total Nasal Symptom Score (TNSS)
Baseline through 2 weeks after randomization

Total Nasal Symptom Score comprised of scoring each of the following symptoms: runny nose, stuffy nose, itchy nose, and sneezing. Each symptom was scored as a 0 (none), 1 (mild), 2 (moderate), or 3 (severe). The 4 individual symptom scores were then added together for a total nasal symptom score. The percent change from baseline was defined as the average of the morning and evening severity scores for the sum of the assessments of the 4 individual scores averaged across all days.

Mean Response at Day 30 to the Patient-rated Relief Assessment Questionnaire
day 30

Mean Patient-Rated Relief Assessment at Day 30. The patient-rated relief assessment (PRRA) was a 4-point scale with 1=Complete Relief; 2=Moderate Relief; 3=Mild Relief; and 4=No Relief.

Daily ocular itching and redness scores
Up to Day 14
Number of Participants With Anatomic Nasal Exam Abnormalities
Day 1 (Baseline) to Exit

The appearance in a participant of any of the following from Baseline: anatomic abnormalities, evidence of infection, bleeding, and/or ulcerations of the mucosa

Peak discomfort score over a 3-minute period after drop instillation
Up to Day 3

Ocular discomfort as measured by Visual Analog Scale (VAS) with 0=none to 50=severe, was assessed by subjects every 30 seconds between 0 to 180 seconds after drop instillation (at 0, 30, 60, 90, 120, 150, and 180 seconds). Peak discomfort (maximum observed VAS discomfort score over the 3-minute period) for each subject in each period was analyzed.

Secondary Endpoints

Mean Subjective Symptoms by Visit
Up to Week 10
Mean Total Redness Score
Day 0 of treatment: 3, 10, 20 minutes post-CAC
Percent Change From Baseline in the Reflective Total Ocular Symptom Score (TOSS)
Baseline through 2 weeks after randomization
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Study Design & Arms

AllocationRANDOMIZED
MaskingSINGLE
ModelPARALLEL
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
PATADAYEXPERIMENTALOlopatadine hydrochloride ophthalmic solution 0.2% in the morning and olopatadine 0.2% vehicle in the evening, 1 drop in each eye for 14 days
PATANOLACTIVE_COMPARATOROlopatadine hydrochloride ophthalmic solution 0.1%, 1 drop in each eye in the morning and evening, for 14 days
AL-4943AEXPERIMENTALOlopatadine Hydrochloride Ophthalmic Solution, 0.2%, 2 drops instilled in each eye twice daily for 10 weeks
Pataday+Pataday VehicleEXPERIMENTALOlopatadine Hydrochloride Ophthalmic Solution 0.2%, 1 drop in 1 eye and Olopatadine 0.2% Vehicle in the contralateral eye
Patanol+Patanol VehicleACTIVE_COMPARATOROlopatadine Hydrochloride Ophthalmic Solution, 0.1%, 1 drop in 1 eye and Olopatadine 0.1% Vehicle in the contralateral eye
Olopatadine 0.6% 1 SprayEXPERIMENTALOlopatadine HCl 0.6% 1 spray per nostril twice daily
Vehicle 1 sprayPLACEBO_COMPARATORVehicle 1 spray per nostril twice daily
Olopatadine 0.6% 2 spraysEXPERIMENTALOlopatadine HCl 0.6% 2 sprays per nostril twice daily
Vehicle 2 spraysPLACEBO_COMPARATORVehicle 2 sprays per nostril twice daily
Olopatadine 0.6% Nasal SprayEXPERIMENTAL2 sprays each nostril twice daily
Placebo Nasal SprayPLACEBO_COMPARATOR2 sprays each nostril twice daily
Olopatadine Hydrochloride 0.2%EXPERIMENTALOlopatadine hydrochloride ophthalmic solution, 0.2%, 1 drop in each eye, once-daily in the morning for 6 weeks
VehiclePLACEBO_COMPARATOROlopatadine hydrochloride ophthalmic solution vehicle, 1 drop in each eye, once-daily in the morning for 6 weeks
1EXPERIMENTALOlopatadine Hydrochloride Nasal Spray 0.6%
2PLACEBO_COMPARATOROlopatadine Hydrochloride Nasal Spray Vehicle
Olopatadine, 0.7%EXPERIMENTALOlopatadine hydrochloride ophthalmic solution, 0.7%, 1 drop instilled in each eye, 1 dose, in Period 1, followed by olopatadine hydrochloride ophthalmic vehicle and ketotifen fumarate ophthalmic solution, 0.025%, Periods 2 and 3, as randomized
ZaditorACTIVE_COMPARATORKetotifen fumarate ophthalmic solution, 0.025%, 1 drop instilled in each eye, 1 dose, in Period 1, followed by olopatadine hydrochloride ophthalmic solution, 0.7% and olopatadine hydrochloride ophthalmic solution vehicle, Periods 2 and 3, as randomized

Interventions

NameTypeDescription
Olopatadine Hydrochloride Ophthalmic Solution 0.2%DRUG -
Olopatadine Hydrochloride Ophthalmic Solution 0.1%DRUG -
Olopatadine 0.2% VehicleDRUGInactive ingredients used as placebo comparator
Olopatadine Hydrochloride Ophthalmic Solution, 0.2%DRUG -
Olopatadine Hydrochloride Ophthalmic Solution, 0.1%DRUG -
Olopatadine 0.1% VehicleDRUGInactive ingredients used as placebo comparator
Olopatadine Hydrochloride Nasal Spray 0.6%DRUGOlopatadine HCl 1 or 2 sprays per nostril twice daily
VehicleDRUGVehicle 1 or 2 sprays per nostril twice daily
Olopatadine 0.6% nasal sprayDRUG2 sprays each nostril twice daily
Placebo Nasal SprayDRUG2 sprays each nostril twice daily
Olopatadine Hydrochloride Ophthalmic Solution VehicleDRUGInactive ingredients used as a placebo comparator
Olopatadine Hydrochloride Nasal Spray VehicleDRUGone spray in each nostril twice daily for 2 weeks
Olopatadine hydrochloride ophthalmic solution, 0.7%DRUGTreatment A
Ketotifen fumarate ophthalmic solution, 0.025%DRUGTreatment C
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Eligibility Criteria

Age Range10 Years to N/A
SexALL
Healthy VolunteersNo

Inclusion Criteria: * Chinese ethnicity; * History of allergic conjunctivitis within the last 2 years; * Positive skin prick test or skin intradermal test documented by a lab report within 24 months of, or at the baseline visit; * Clinical diagnosis of allergic conjunctivitis with specific signs an...

Countries:JapanUnited States
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Frequently asked questions about Olopatadine, 0.7%

What is Olopatadine 0.2% used for?

Olopatadine 0.2% is used for allergic rhinitis, seasonal allergic rhinitis, perennial allergic rhinitis, and allergic conjunctivitis. It is an ophthalmic small molecule being developed by Alcon Inc. for these allergic conditions.

Who makes Olopatadine 0.2%?

Olopatadine 0.2% is developed by Alcon Inc., a company traded under the ticker ALC. Alcon is conducting clinical trials to evaluate the safety and efficacy of this drug for allergic rhinitis and allergic conjunctivitis.

What phase is Olopatadine 0.2% in?

Olopatadine 0.2% is in Phase 3 clinical development. It is an investigational drug, meaning it has not been approved by regulatory authorities. The Phase 3 trials are completed and include studies for perennial allergic rhinitis, seasonal allergic rhinitis, and allergic conjunctivitis.

What clinical trials is Olopatadine 0.2% in?

Olopatadine 0.2% has completed several clinical trials, including NCT00578331 for perennial allergic rhinitis, NCT00578929 for seasonal allergic rhinitis, and NCT02322216 for allergic conjunctivitis. These trials enrolled a total of 2,388 participants across the United States and other regions.

Is Olopatadine 0.2% the same as Patanase?

Olopatadine 0.2% is related to Patanase, as both contain olopatadine. However, Olopatadine 0.2% is an ophthalmic solution, while Patanase is a nasal spray. They are used for different routes of administration in treating allergic conditions.