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Temodar and O6-Benzylguanine

Phase 2

Glioblastoma Multiforme | Small molecule | Oncology |Akebia Therapeutics, Inc.|Last Updated: Jul 9, 2014

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
ACTIVE_CONTROLLEDDMCBiomarker
Total Trials1
Total Enrollment67
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT00613093Ph. II Temozolomide + O6-BG in Treatment of Pts w Temozolomide-Resistant Malignant GliomaPHASE2 COMPLETED 67Oct 1, 2002Aug 1, 2008Jul 9, 20141 United States
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Study Endpoints
Primary Endpoints
Radiographic evidence of tumor response
6 months
Secondary Endpoints
6 month progression-free survival
6 months
Relationship between tumor AGT at original diagnosis & response to Temozolomide + O6-BG
6 months
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Patients with glioblastoma multiformeACTIVE_COMPARATOR -
Patients with Anaplastic GliomaACTIVE_COMPARATOR -
Interventions
NameTypeDescription
Temodar and O6-Benzylguanine (BG)DRUGObjectives of study are to define role of BG in restoring Temodar sensitivity in patients with Temodar-resistant malignant glioma and to further define the toxicity of combination therapy using Temodar + BG. 2 separate strata accrued independently of each other: Stratum 1-patients with glioblastoma multiforme (GBM). Stratum 2-patients with anaplastic glioma (AG). BG at 120mg/m2 administered intravenously over 1 hour followed immediately by 48-hour infusion at 30mg/m2/24 hours. Temodar 472mg/m2 administered orally, in fasting state, within 60 minutes of end of the 1-hour administration of BG infusion. Treatment cycles may be repeated every 28 days following dose of Temodar from previous cycle.
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Eligibility Criteria
Age Range18 Years — N/A
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: * Patients have recurrent/progressive Malignant Glioma (MG). Stereotactic biopsy at time of recurrence/progression is only required if radiation-induced necrosis is suspected * Patients have MG resistant to Temodar, which is defined as \> or = to 25 percent increase in tumor gro...

Countries:United States
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