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Clarithromycin

Phase 1

Helicobacter Pylori | Small molecule | Gastrointestinal |Takeda Pharmaceutical Company Limited|Last Updated: Sep 19, 2024

Success Probability

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Market & Valuation

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Trial Design

RandomizedDouble-BlindACTIVE_CONTROLLED
Total Trials2
Total Enrollment74

FDA Designations

No designations recorded

Clinical trial landscape

Clarithromycin · 3 trials · 2 indications

Phase 1 3
NCT02542657Ixazomib with Pomalidomide, Clarithromycin and Dexamethasone in Treating Patients with Multiple MyelomaMyeloma
ACTIVE NOT_RECRUITING30 Analytics
NCT04753437A Study of Vonoprazan in Adults With Helicobacter PyloriHelicobacter Pylori
COMPLETED44 Analytics
NCT02892409TAK-438 Bismuth Drug Interaction StudyHelicobacter Pylori
COMPLETED30 Analytics
PHASE1ACTIVE NOT_RECRUITING
Ixazomib with Pomalidomide, Clarithromycin and Dexamethasone in Treating Patients with Multiple Myeloma
MyelomaUnlock trial analytics
PHASE1COMPLETED
A Study of Vonoprazan in Adults With Helicobacter Pylori
Helicobacter PyloriUnlock trial analytics
PHASE1COMPLETED
TAK-438 Bismuth Drug Interaction Study
Helicobacter PyloriUnlock trial analytics

Study Endpoints

Primary Endpoints

MTD of clarithromycin when given in combination with ixazomib citrate, pomalidomide, and dexamethasone assessed by the National Cancer Institute (NCI) Common Terminology Criteria for Adverse Events (CTCAE) version 4.0 (Phase I)
28 days

The MTD is defined as the highest dose tested in which fewer than 33% of patients experience a dose limiting toxicity and at least 6 patients have been treated at that dose. The MTD will be the recommended Phase 2 dose, provided that other safety considerations are acceptable.

Cmax: Maximum Observed Plasma Concentration for Bismuth
Day 14: 0 to 12 hours after the morning dose
AUCτ: Area Under the Plasma Concentration-time Curve During a Dosing Interval τ for Bismuth
Day 14: 0 to 12 hours after the morning dose
Aeτ: Total Amount of Bismuth Excreted in Urine During a Dosing Interval τ for Bismuth
Day 14: 0 to 12 hours after the morning dose
Percentage of Participants Who Experience at Least One Treatment Emergent Adverse Event (TEAE)
Baseline up to Day 17
Percentage of Participants Who Discontinue Due to an Adverse Event (AE)
Baseline up to Day 17
Percentage of Participants Who Meet the Markedly Abnormal Criteria for Safety Laboratory Tests at Least Once Post-dose
Baseline up Day 15
Percentage of Participants Who Meet the Markedly Abnormal Criteria for Vital Sign Measurements at Least Once Post-dose
Baseline up to Day 15
Percentage of Participants Who Meet the Markedly Abnormal Criteria for Safety Electrocardiogram (ECG) Parameters at Least Once Post-dose
Baseline up to Day 15
AUCτ: Area Under the Plasma Concentration-time Curve From Time 0 to Time Tau Over the Dosing Interval for Bismuth
Day 14 pre-dose and at multiple timepoints (up to 12 hours) post-dose
Aeτ: Amount of Drug Excreted in Urine During a Dosing Interval for Bismuth
Day 14 pre-dose and at multiple timepoints (up to 12 hours) post-dose

Secondary Endpoints

Clinical best response
Up to 3 years
Percentage of Participants Who Experience at Least One Treatment-Emergent Adverse Event (TEAE)
From the first dose of study drug up to Day 17
Percentage of Participants Who Discontinued Study Drug Due to a Treatment-Emergent Adverse Event (TEAE)
From the first dose of study drug up to Day 17
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Study Design & Arms

AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT

Treatment Arms

ArmTypeDescription
Treatment (PiC-D therapy)EXPERIMENTALPatients receive pomalidomide PO QD on days 1-21; ixazomib citrate PO on days 1, 8, and 15; clarithromycin PO BID on days 15-21 of course 1 and days 1-21 of courses 2-6; and dexamethasone PO on days 1, 8, 15, and 22. Treatment repeats every 28 days for 6 courses in the absence of disease progression or unacceptable toxicity. MAINTENANCE THERAPY: Patients receive pomalidomide, ixazomib citrate, and dexamethasone as above and receive clarithromycin PO BID or QD. Courses repeat every 28 days in the absence of disease progression or unacceptable toxicity.
Clarithromycin + Amoxicillin + Bismuth + VonoprazanEXPERIMENTALClarithromycin 500 milligram (mg), tablets, orally, BID, along with amoxicillin 1000 mg, capsules, orally, BID, bismuth potassium citrate 600 mg, capsules, orally, BID, and vonoprazan 20 mg, tablets, orally, BID on Days 1 to 14.
Clarithromycin + Amoxicillin + Bismuth + EsomeprazoleACTIVE_COMPARATORClarithromycin 500 mg, tablets, orally, BID, along with amoxicillin 1000 mg, capsules, orally, BID, bismuth potassium citrate 600 mg, capsules, orally, BID, and esomeprazole 20 mg, tablets, orally, BID on Days 1 to 14.
Clarithromycin + Amoxicillin + Bismuth + LansoprazoleACTIVE_COMPARATORClarithromycin 500 milligram (mg), tablets, orally, twice daily, along with amoxicillin 1000 mg capsules, orally, twice daily, tripotassium bismuth dicitrate 600 mg, tablets, orally, twice daily, and lansoprazole 30 mg, capsules, orally, twice daily on Days 1 to 14.
Clarithromycin + Amoxicillin + Bismuth + TAK-438EXPERIMENTALClarithromycin 500 mg, tablets, orally, twice daily, along with amoxicillin 1000 mg, capsules, orally, twice daily, tripotassium bismuth dicitrate 600 mg, tablets, orally, twice daily, and TAK-438 20 mg, tablets, orally, twice daily on Days 1 to 14.

Interventions

NameTypeDescription
ClarithromycinDRUGGiven PO
DexamethasoneDRUGGiven PO
Ixazomib CitrateDRUGGiven PO
PomalidomideDRUGGiven PO
AmoxicillinDRUGAmoxicillin capsules.
Bismuth potassium citrateDRUGBismuth potassium citrate tablets.
EsomeprazoleDRUGEsomeprazole tablets.
VonoprazanDRUGVonoprazan tablets.
Tripotassium bismuth dicitrateDRUGTripotassium bismuth dicitrate tablets
LansoprazoleDRUGLansoprazole capsules
TAK-438DRUGTAK-438 tablets
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Eligibility Criteria

Age Range18 Years to N/A
SexALL
Healthy VolunteersNo
Study Sites3

Inclusion Criteria: * Voluntary written consent * Patients must have a confirmed biopsy diagnosis of a multiple myeloma * Submission of original biopsy for review and verification by hematopathologist at local institution * Patients must have measurable disease according to International Myeloma Wo...

Countries:United StatesChinaSouth Korea
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Frequently asked questions about Clarithromycin

What is Clarithromycin used for?

Clarithromycin is a small molecule being studied for use in myeloma and Helicobacter pylori infection. In clinical trials, it is being evaluated as part of combination therapy for multiple myeloma and in drug interaction studies related to Helicobacter pylori treatment. It is currently in Phase 1 clinical development.

What does Clarithromycin target?

Clarithromycin is a macrolide antibiotic that works by inhibiting bacterial protein synthesis. It binds to the 50S ribosomal subunit of susceptible bacteria, blocking peptide bond formation and thereby stopping bacterial growth. This mechanism underlies its use in treating Helicobacter pylori infections.

Who makes Clarithromycin?

Clarithromycin is being developed by Takeda Pharmaceutical Company Limited, which trades under the ticker TAK. Takeda is conducting clinical trials to evaluate the drug for multiple myeloma and Helicobacter pylori infections.

What phase is Clarithromycin in?

Clarithromycin is in Phase 1 clinical development. It is an investigational drug and has not been approved by regulatory authorities for the indications being studied. The ongoing Phase 1 trial is active but not recruiting patients.

What clinical trials is Clarithromycin in?

Clarithromycin is involved in three clinical trials. NCT02542657 is a Phase 1 study combining ixazomib, pomalidomide, clarithromycin, and dexamethasone for multiple myeloma. NCT02892409 and NCT04753437 are Phase 1 studies related to Helicobacter pylori, including a drug interaction study and a vonoprazan study.

Is Clarithromycin the same as TAK-438?

No, Clarithromycin is not the same as TAK-438. TAK-438 is a separate drug being studied in combination with clarithromycin for Helicobacter pylori infection. Clarithromycin is the antibiotic component, while TAK-438 is a potassium-competitive acid blocker.