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TVB-2640 -

Phase 1

Non-alcoholic Steatohepatitis | Small molecule | Infectious Disease |Sagimet Biosciences Inc. - Series A|Last Updated: Dec 26, 2023

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment48
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT05835180A Phase I Pharmacokinetic Study of TVB-2640 (Denifanstat) in Subjects With Mild, Moderate, or Severe Hepatic Impairment Compared to Subjects With Normal Hepatic FunctionPHASE1 COMPLETED 48May 1, 2023Dec 18, 2023Dec 26, 20233 United States, Hungary
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Study Endpoints
Primary Endpoints
Total TVB-2640 plasma concentration-time (AUC) at steady state
Day 4

Total TVB-2640 plasma concentration-time curve during a dosing interval at steady-state

Unbound TVB-2640 plasma concentration-time (AUC) at steady state
Day 4

Unbound TVB-2640 plasma concentration-time curve during a dosing interval at steady-state

Maximum plasma concentration (Cmax) for total TVB-2640 at steady state
Day 4
Maximum plasma concentration (Cmax) for unbound TVB-2640 at steady state
Day 4
incidence and severity of AEs
Screening to Day 7
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
TVB-2640 50 mg - normal hepatic functionEXPERIMENTALHealthy subjects with normal hepatic function receive 50 mg PO daily from Day 1 to Day 4
TVB-2640 50 mg - mild hepatic functionEXPERIMENTALSubjects with mild hepatic impairment will receive 50 mg PO daily from Day 1 to Day 4
TVB-2640 50 mg - moderate hepatic functionEXPERIMENTALSubjects with moderate hepatic impairment will receive 50 mg PO daily from Day 1 to Day 4
TVB-2640 50 mg - severe hepatic functionEXPERIMENTALSubjects with severe hepatic impairment will receive 50 mg PO daily from Day 1 to Day 4
Interventions
NameTypeDescription
TVB-2640 - 50 mgDRUGTVB-2640 -50 mg administered orally once daily
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Eligibility Criteria
Age Range18 Years — 75 Years
SexALL
Healthy VolunteersYes
Study Sites3

Key Inclusion Criteria: Subjects must satisfy all of the following criteria at the Screening visit unless otherwise stated: All Subjects * Males or females, of any race, between 18 and 75 years of age, inclusive. * Body mass index between 18.0 and 42.0/45.0 kg/m2 (inclusive; up to 42.0 kg/m2 for ...

Countries:United StatesHungary
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