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dacomitinib fasted

Phase 1

Healthy Volunteers | Small molecule | Other |Pfizer, Inc.|Last Updated: Dec 18, 2013

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedCONTROLLED
Total Trials1
Total Enrollment24
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01702506Evaluation Of The Potential Effect That The Administration Of Food Or Antacid Medication May Have In The Oral Absorption Of Dacomitinib (PF-00299804)PHASE1 COMPLETED 24Oct 1, 2012Jan 1, 2013Dec 18, 20131 Belgium
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Study Endpoints
Primary Endpoints
Area Under the Curve From Time Zero to Extrapolated Infinite Time [AUC (0 - 8)]
2 weeks

AUC (0 - 8)= Area under the plasma concentration versus time curve (AUC) from time zero (pre-dose) to extrapolated infinite time (0 - 8). It is obtained from AUC (0 - t) plus AUC (t - 8). For dacomitinib and PF-05199265

Maximum Observed Plasma Concentration (Cmax)
2 weeks

For dacomitinib and PF-05199265

Secondary Endpoints
Area Under the Curve From Time Zero to Last Quantifiable Concentration [AUC (0-t)]
2 weeks
Area under the Concentration-Time Curve (AUC)
3 days
Apparent Oral Clearance (CL/F)
2 weeks
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
FastedEXPERIMENTALDacomitinib administered under fasted conditions
FedEXPERIMENTALDacomitinib administered under fed conditions
AntacidEXPERIMENTALDacomitinib administered under antacid treatment
Interventions
NameTypeDescription
dacomitinib fastedDRUGOvernight fasted subjects will receive a single 45 mg dose of dacomitinib
dacomitinib fedDRUGSubjects will receive a single 45 mg dose of dacomitinib with a high calorie high fat meal
dacomitinib+antacidDRUGSubjects will receive a single 45 mg dose of dacomitinib when there are treated with rabeprazole
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy subjects including males between the ages of 18 and 55 years. Females of non childbearing potential . * Body Mass Index (BMI) of 17.5 to 30.5 kg/m2; and a total body weight \>50 kg (110 lbs). * An informed consent document signed and dated by the subject. Exclusion Cr...

Countries:Belgium
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