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PF-06882961,

Phase 1

Healthy Volunteer | Small molecule | Other |Pfizer, Inc.|Last Updated: Nov 25, 2020

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLED
Total Trials1
Total Enrollment6
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04495140Study To Characterize Mass Balance, Absolute Bioavailability, Fraction Absorbed And Pharmacokinetics Of 14C PF-06882961PHASE1 COMPLETED 6Jul 22, 2020Oct 15, 2020Nov 25, 20202 Netherlands
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Study Endpoints
Primary Endpoints
Total recovery of radioactivity in urine and feces, following oral administration of [14C] PF-06882961 in period 1
Baseline through approximately hour 312 (day 14). Period 1 is 14 days

Total recovery of radioactivity in urine and feces, and both routes combined, expressed as a percent of total oral radioactive dose administered.

Secondary Endpoints
Metabolite profiling/identification in plasma, urine, and feces
0, 0.5, 1, 2, 3, 4, 6, 9, 12, 16, 24, 36, 48, 72, 96-312 hour (hr)
Plasma Cmax to describe plasma PK of total radioactivity following administration of single, oral dose of [14C] PF-06882961
0, 0.5, 1, 2, 3, 4, 6, 9, 12, 16, 24, 36, 48, 72, 96 hr
Plasma Tmax to describe the PK of total radioactivity following administration of single, oral dose of [14C]PF-06882961
0, 0.5, 1, 2, 3, 4, 6, 9, 12, 16, 24, 36, 48, 72, 96 hr
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
Oral [14C]PF-06882961, 50 mgEXPERIMENTALIn this arm, a single oral dose of \[14C\]PF-06882961, 50 mg will be administered as a liquid formulation.
Oral PF-06882961 50 mg and intravenous [14C]PF-06882961 100 ugEXPERIMENTALIn this arm, single oral dose of unlabeled PF-06882961, 50 mg will be administered as a liquid formulation. Approximately 3 hours after the administration of the unlabeled oral dose, a single dose of \[14C\]PF-06882961, 100 ug, will be administered via intravenous infusion.
Interventions
NameTypeDescription
[14C]PF-06882961, 50 mgDRUGA single oral dose of \[14C\]PF-06882961, will be administered as a liquid formulation.
PF-06882961, 50 mg and [14C]PF-06882961, 100 ugDRUGA single, oral, unlabeled dose of PF-06882961, 50 mg will be administered as a liquid formulation. Approximately 3 hours after the administration of the unlabeled oral dose, a single dose of \[14C\]PF-06882961 will be administered via intravenous infusion.
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Eligibility Criteria
Age Range18 Years — 54 Years
SexMALE
Healthy VolunteersYes
Study Sites2

Inclusion Criteria: * Male participants between 18 to 54 years of age * Healthy and capable of signing informed consent document * Willing to comply to all scheduled visits, lab tests, lifestyle considerations and study procedures * Body mass index (BMI) of 17.5 to 30 kg/m2; and a total body weight...

Countries:Netherlands
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