Recent Updates
Recently added Catalysts

Trametinib

Phase 1

KRAS Mutation-Related Tumors | Small molecule | Oncology |BeOne Medicines Ltd.|Last Updated: Jun 13, 2024

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
UNCONTROLLEDBiomarker
Total Trials1
Total Enrollment60
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT06456138Trametinib Plus Anlotinib Combined With Tislelizumab in KRAS-mutant NSCLCPHASE1 NOT YET_RECRUITING 60Jul 1, 2024Dec 31, 2028Jun 13, 20241 China
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
RP2D
up to 12 months

recommended phase 2 dose

PFS
up to 18 months

progression-free survival

Secondary Endpoints
ORR
up to 12 months
OS
up to 24 months
DOR
up to 18 months
Unlock Study Endpoints
Study Design & Arms
AllocationNA
MaskingNONE
ModelSINGLE_GROUP
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Trametinib + Anlotinib + TislelizumabEXPERIMENTALIn Phase I, there are four treatment arms: anlotinib (6 mg) plus trametinib (1 mg) plus tislelizumab (200 mg, Q3W), anlotinib (6 mg) plus trametinib (2 mg) plus tislelizumab (200 mg, Q3W), anlotinib (8 mg) plus trametinib (1 mg) plus tislelizumab (200 mg, Q3W), and anlotinib (8 mg) plus trametinib (2 mg) plus tislelizumab (200 mg, Q3W). In Phase II, there is one treatment arm including trametinib (RP2D) plus anlotinib (RP2D) plus tislelizumab (200 mg, Q3W).
Interventions
NameTypeDescription
TrametinibDRUGTrametinib will be administrated orally every day.
AnlotinibDRUGAnlotinib will be administrated orally from day 1 to day 14 per 21-day cycle.
TislelizumabDRUGTislelizumab will be administered at full dose (200mg, Q3W) on the patient who received the efficacy evaluation of stable disease (SD) or partial response (PR) or complete response (CR) after 2 cycles' treatment of trametinib plus anlotinib.
Unlock Study Design Details
Eligibility Criteria
Age Range18 Years — 75 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: 1. According to the 8th edition of the AJCC/UICC TNM staging system for NSCLC, patients with locally advanced (stage III B/III C), metastatic or recurrent (stage IV) NSCLC confirmed by histology or cytology who are unable to undergo surgery and radical concomitant radiochemother...

Countries:China
Unlock Eligibility Criteria
Recent Changes (Last 90 Days)
LOWMay 24, 2026NCT06456138studyFirstPostDate: changed