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Part A: RPL554

Phase 2

Pulmonary Disease, Chronic Obstructive | Small molecule | Other |Merck & Company, Inc.|Last Updated: Sep 26, 2022

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindACTIVE_CONTROLLEDBiomarker
Total Trials1
Total Enrollment37
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04027439Study Evaluating 5 Doses of RPL554 and Placebo in COPD Patients Via a Dry Powder InhalerPHASE2 COMPLETED 37Dec 10, 2018May 23, 2019Sep 26, 20221 United States
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Study Endpoints
Primary Endpoints
Part A: RPL554 Plasma Pharmacokinetic Parameter (AUC0-12)
Day 1

RPL554 Plasma pharmacokinetics AUC0-12 (Area under the Curve) after single dose

Part A: RPL554 Plasma Pharmacokinetic Parameter (AUC 0-t)
Day 1

RPL554 Area under the curve at maximum concentration after a single dose

Part A: RPL554 Plasma Pharmacokinetic Parameter (Half-life)
Day 1

RPL554 Plasma pharmacokinetics Half-life concentration after a single dose

Part B: Change From Baseline in Peak FEV1 (Over 4 Hours)
Day 7

Change from Baseline FEV1 to Peak FEV1 (over 4 hours) on Day 7

Secondary Endpoints
Part A: Change From Baseline in Average FEV1 (Over 4 Hours)
Day 1
Part A: Change From Baseline in Average FEV1 (Over 12 Hours)
Day 1
Part A: Change From Baseline in Peak FEV1 (Over 4 Hours)
Day 1
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelFACTORIAL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part A: RPL554ACTIVE_COMPARATORPlacebo controlled, parallel group single dose. Five of the 6 treatment arms will be double-blind and one will be single-blind
Part B: RPL554ACTIVE_COMPARATORDouble-blind, placebo-controlled, complete block cross-over
Interventions
NameTypeDescription
Part A: RPL554DRUG1 dose of either 50mcg/100mcg/1500mcg/3000mcg/6000mcg or placebo via dry powder inhaler
Part B: RPL554DRUGPatients will receive 4 or 5 repeat dose treatments in crossover fashion - doses will be confirmed after Part A
PlacebosDRUGPart A: 1 dose of either 50ncg/100ncg/1500ncg/3000ncg/6000ncg or placebo via dry powder inhaler. Part B: Patients will receive 4 or 5 repeat dose treatments in crossover fashion - doses will be confirmed after Part A.
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Eligibility Criteria
Age Range40 Years — 80 Years
SexALL
Healthy VolunteersNo
Study Sites1

Inclusion Criteria: 1. Sign an informed consent document indicating they understand the purpose of and procedures required for the study and are willing to participate in the study. 2. For males, not to donate sperm and either be sexually abstinent or use contraception as specified by the protocol....

Countries:United States
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