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JNJ-42165279 2.5 -

Phase 1

Healthy Volunteers | Small molecule | Other |Johnson & Johnson|Last Updated: Jul 6, 2017

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindCONTROLLED
Total Trials1
Total Enrollment29
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01650597A Single Ascending Dose Study to Investigate the Safety, Tolerability, and Pharmacokinetics of JNJ-42165279 in Healthy Male ParticipantsPHASE1 COMPLETED 29Aug 1, 2011May 1, 2012Jul 6, 20171 Belgium
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Study Endpoints
Primary Endpoints
Incidents of adverse events amongst participants (Part 1)
Day -21 to Day 114 (~19 wks)

As a measure of safety.

Incidents of adverse events amongst participants (Part 2)
Day -21 to Day 23 (~6 wks)
Pharmacokinetics of JNJ-42165279 as measured by Cmax (Part 1)
Day 1 to Day 4

Cmax is defined as maximum plasma concentration of JNJ-42165279.

Pharmacokinetics of JNJ-42165279 as measured by Cmax (Part 2)
Day 1 to Day 7
Pharmacokinetics of JNJ-42165279 as measured by AUC (Part 1)
Day 1 to Day 4

AUC is defined area under the plasma concentration time curve from 0 to t hours post dosing of JNJ-42165279.

Pharmacokinetics of JNJ-42165279 as measured by AUC (Part 2)
Day 1 to Day 7
Secondary Endpoints
Fatty acid amide hydrolase (FAAH) inhibition in white blood cells (WBCs) (Part 1)
Day 1 to Day 4
FAAH inhibition in WBC (Part 2)
Day 1 to Day 7 and Day 9
Effects on mood (Part 1)
Day 1 and Day 2
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Study Design & Arms
AllocationRANDOMIZED
MaskingDOUBLE
ModelCROSSOVER
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
Part 1 - Panel 1EXPERIMENTALThe participants will receive 3 or 4 ascending doses (2.5, 10, 30, 100, 250, 500 mg) of JNJ-42165279 and placebo during the study.
Part 1 - Panel 2EXPERIMENTALThe participants will receive 3 or 4 ascending doses (2.5, 10, 30, 100, 250, 500 mg) of JNJ-42165279 and placebo during the study.
Part 2 (parallel)- additional cohortEXPERIMENTALThe participants will receive repeated daily dosing of 100 mg JNJ-42165279 or placebo for 6 consecutive days.
Interventions
NameTypeDescription
JNJ-42165279 2.5 - 500 mg oralDRUGType=exact number, unit=mg, numbers=2.5, 10, 30, 100, 250 and 500, form=suspension, route=oral use. One single dose administered orally.
PlaceboDRUGType=exact number, unit=mg, form=solution, route=oral use. One single dose administered orally.
JNJ-42165279 100 mg oralDRUGType=exact number, unit=mg, form=solution, route=oral use. One single dose administered orally.
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Eligibility Criteria
Age Range18 Years — 55 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Has a body mass index between 18 and 30 kg/m2 and body weight not less than 50 kg. * Must adhere to required contraception (subject and partner, if applicable) during the study and for 3 months after study * Must agree to not donate sperm during the study and for 3 months afte...

Countries:Belgium
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