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abacavir /lamivudine

Phase 1

Healthy Subjects | Small molecule | Other |GSK plc|Last Updated: Aug 8, 2011

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedUNCONTROLLEDBiomarker
Total Trials1
Total Enrollment18
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01366547Relative Bioavailability Study of Two New Dolutegravir/Abacavir/Lamivudine Fixed Dose Combination TabletsPHASE1 COMPLETED 18Jun 1, 2011Jul 1, 2011Aug 8, 20111 United States
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Study Endpoints
Primary Endpoints
Plasma DTG AUC(0-infinity)
48 hours post dose
Plasma ABC AUC(0-infinity)
48 hours post dose
Plasma 3TC AUC(0-infinity)
48 hours post dose
Plasma DTG AUC(0-t)
48 hours post dose
Plasma ABC AUC(0-t)
48 hours post dose
Plasma 3TC AUC(0-t)
48 hours post dose
Plasma DTG Cmax
48 hours post dose
Plasma ABC Cmax
48 hours post dose
Plasma 3TC Cmax
48 hours post dose
Secondary Endpoints
Change from baseline in 12-lead ECG
48 hours post dose
Plasma DTG tlag
48 hours post dose
Number of subjects with adverse events
48 hours post dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
Treatment Arms
ArmTypeDescription
Single ArmEXPERIMENTALSubjects will be randomized in a three-way crossover design to receive a single dose of each of two different tablet formulations of dolutegravir 50 mg/abacavir 600 mg/lamivudine 300 mg or dolutegravir 50 mg plus EPZICOM (abacavir 600mg/lamivudine 300 mg). There will be a screening visit within 30 days prior to first dose and a follow-up visit 7-14 days after the last dose.
Interventions
NameTypeDescription
Dolutegravir 50 mg/abacavir 600 mg/lamivudine 300 mgDRUGDolutegravir 50 mg/abacavir 600 mg/lamivudine 300 mg is an experimental fixed dose combination tablet of an experimental integrase inhibitor (dolutegravir) and two FDA approved nucleoside reverse transcriptase inhibitors (abacavir and lamivudine)
Dolutegravir 50 mgDRUGDolutegravir is an experimental drug in the integrase inhibitor class that is being studied for the treatment of HIV infection.
abacavir 600 mg/lamivudine 300 mgDRUGThis is an FDA approved fixed dose combination tablet of two nucleoside reverse transcriptase inhibitors
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Eligibility Criteria
Age Range18 Years — 65 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy as determined by a responsible and experienced physician, based on a medical evaluation including medical history, physical examination, laboratory tests and cardiac monitoring. * Male or female between 18 and 65 years of age inclusive, at the time of signing the infor...

Countries:United States
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