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Pirfenidone

Phase 1

Healthy | Small molecule | Other |Galapagos NV|Last Updated: Sep 19, 2024

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLED
Total Trials1
Total Enrollment58
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04971746Drug-drug Interaction Study with GLPG4716 and Nintedanib and Pirfenidone in Healthy SubjectsPHASE1 COMPLETED 58Jul 19, 2021May 9, 2022Sep 19, 20241 Germany
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Study Endpoints
Primary Endpoints
Maximum observed plasma concentration (Cmax) of pirfenidone
From Day 1 pre-dose until Day 15

To determine the effect of GLPG4716 on the PK of pirfenidone

Area under the plasma concentration-time curve from time zero to infinity (AUC0-inf) of pirfenidone
From Day 1 pre-dose until Day 15

To determine the effect of GLPG4716 on the PK of pirfenidone

Cmax of nintedanib
From Day 1 pre-dose until Day 15

To determine the effect of GLPG4716 on the PK of nintedanib.

AUC0-inf of nintedanib
From Day 1 pre-dose until Day 15

To determine the effect of GLPG4716 on the PK of nintedanib.

Secondary Endpoints
Frequency and severity of treatment-emergent adverse events (TEAEs), treatment-emergent serious adverse events (SAEs), and TEAEs leading to treatment discontinuations.
From Day 1 through study completion, an average of 2 months
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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
GLPG4716 and pirfenidoneEXPERIMENTAL -
GLPG4716 and nintedanibEXPERIMENTAL -
Interventions
NameTypeDescription
PirfenidoneDRUGOn Days 1 and 13, participants will receive an oral dose of pirfenidone.
GLPG4716DRUGFrom Day 3 to Day 14, participants will receive GLPG4716 daily.
NintedanibDRUGOn Days 1 and 13, participants will receive an oral dose of nintedanib.
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Male or female between 18 and 55 years of age (extremes included), on the date of signing the informed consent form (ICF). Female subjects should be of non-childbearing potential. * A body mass index (BMI) between 18.0 and 30.0 kg/m2, inclusive. * Judged to be in good health b...

Countries:Germany
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