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GLPG3312 IR

Phase 1

Healthy | Small molecule | Other |Galapagos NV|Last Updated: Mar 19, 2020

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment95
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03800472A Study Investigating the Safety, Absorption and Elimination of GLPG3312, a New Drug in the Treatment of Inflammatory DiseasesPHASE1 COMPLETED 95Jan 15, 2019Mar 10, 2020Mar 19, 20201 Netherlands
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Study Endpoints
Primary Endpoints
Frequency and severity of treatment emergent adverse events (TEAEs), treatment-emergent serious adverse events, and TEAEs leading to treatment discontinuations
From screening through study completion, an average of 9 months.

To evaluate the safety and tolerability of oral single and multiple ascending doses of GLPG3312, in adult, healthy, subjects, when given as Immediate Release (IR) formulation (in fasted conditions) or as Modified Release (MR) formulation (in fasted and fed conditions)

Secondary Endpoints
Maximum observed plasma concentration (Cmax) of GLPG3312 (μg/mL) (Part 1)
Between Day 1 pre-dose and Day 4
Maximum observed plasma concentration (Cmax) of GLPG3312 (μg/mL) (Part 2)
Between Day 1 pre-dose and Day 7
Maximum observed plasma concentration (Cmax) of GLPG3312 (μg/mL) under fed conditions (high-fat high calorie) versus fasted conditions (Part 3)
Between Day 1 pre-dose and Day 7
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
GLPG3312 SAD IR (Part 1)EXPERIMENTALSingle doses of GLPG3312 IR
Placebo SAD IR (Part 1)PLACEBO_COMPARATORSingle doses of Placebo IR
GLPG3312 SAD MR (Part 2)EXPERIMENTALSingle doses of GLPG3312 MR
Placebo SAD MR (Part 2)PLACEBO_COMPARATORSingle doses of Placebo MR
GLPG3312 FE MR (Part 3)EXPERIMENTALSingle dose of GLPG3312 MR in fed and fasted state
GLPG3312 MAD MR (Part 4)EXPERIMENTALMultiple doses of GLPG3312 MR
Placebo MAD MR (Part 4)PLACEBO_COMPARATORMultiple doses of Placebo MR
GLPG3312 MAD MR optimized (Part 4)EXPERIMENTALMultiple doses of GLPG3312 MR
Placebo MAD MR optimized (Part 4)PLACEBO_COMPARATORMultiple doses of Placebo MR
Interventions
NameTypeDescription
GLPG3312 IRDRUGGLPG3312 IR tablets, up to 4 single ascending oral doses (A, B, C, D).
PlaceboDRUGPlacebo tablets
GLPG3312 MRDRUGGLPG3312 MR film-coated tablets, up to 4 single ascending oral doses (H, I, J, K).
GLPG3312 FE MRDRUGGLPG3312 MR film-coated tablets, single oral dose (N) on 2 occasions, i.e. in fed state after a high-fat high-calorie breakfast, and in fasted state.
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Eligibility Criteria
Age Range18 Years — 55 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Male or female between 18 to 55 years of age (extremes included), on the date of signing the Informed Consent Form (ICF). Female should be of non-childbearing potential defined as permanently surgically sterile (bilateral oophorectomy, i.e. surgical removal of ovaries, bilater...

Countries:Netherlands
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