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GLPG3067 single dose

Phase 1

Healthy | Small molecule | Other |Galapagos NV|Last Updated: Apr 10, 2018

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDBiomarker
Total Trials1
Total Enrollment81
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03128606A Study to Assess Safety, Tolerability and Pharmacokinetics of GLPG3067 in Healthy Subjects.PHASE1 COMPLETED 81Mar 28, 2017Feb 20, 2018Apr 10, 20181 Belgium
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Study Endpoints
Primary Endpoints
Change versus placebo in the proportion of subjects with adverse events
Between screening and 14 days after the last dose

To assess safety and tolerability of single ascending doses, multiple ascending doses of GLPG3067 alone, or in combination with GLPG2222, or in combination with GLPG2222 and GLPG2737 versus placebo in healthy subjects

Secondary Endpoints
Maximum observed plasma concentration of GLPG3067 (Cmax) given alone or in combination with GLPG2222 or in combination with GLPG2222 and GLPG2737
Between Day 1 predose and 10 days after the last dose
Area under the plasma concentration-time curve of GLPG3067 (AUC0-t) given alone or in combination with GLPG2222 or in combination with GLPG2222 and GLPG2737
Between Day 1 predose and 10 days after the last dose
Ratio of 4-beta-hydroxycholesterol/cholesterol in plasma after multiple oral doses in healthy subjects
Day 1 predose and Day 14
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelSEQUENTIAL
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
GLPG3067 single doseEXPERIMENTALSingle dose of GLPG3067 oral suspension at up to 6 dose levels in ascending order.
Placebo single dosePLACEBO_COMPARATORSingle dose of Placebo oral suspension.
GLPG3067 oral suspension fed 1EXPERIMENTALSingle dose 1 of GLPG3067 oral suspension after a standardized breakfast.
GLPG3067 oral tablet fed 1EXPERIMENTALSingle dose 1 of GLPG3067 oral tablet after a standardized breakfast.
GLPG3067 oral tablet fasted 1EXPERIMENTALSingle dose 1 of GLPG3067 oral tablet after an overnight fast.
GLPG3067 oral tablet fed 2EXPERIMENTALSingle dose 2 of GLPG3067 oral tablet after a standardized breakfast.
GLPG3067 oral tablet fed 2 high-fat high-calorieEXPERIMENTALSingle dose 2 of GLPG3067 oral tablet after a high-fat high-calorie breakfast
GLPG3067 multiple doseEXPERIMENTALMultiple doses of GLPG3067 oral suspension at up to 5 dose levels in ascending order.
Placebo multiple dosePLACEBO_COMPARATORMultiple doses of Placebo oral suspension.
GLPG3067/GLPG2222 multiple doseEXPERIMENTALMultiple doses of GLPG3067 oral suspension combined with GLPG2222 oral tablet up to 2 dose levels in ascending order.
GLPG3067/GLPG2222 Placebo multiple dosePLACEBO_COMPARATORMultiple doses of GLPG3067 matching placebo oral suspension combined with GLPG2222 matching placebo oral tablet.
GLPG3067/GLPG2222/GLPG2737 multiple doseEXPERIMENTALMultiple doses of GLPG3067 oral tablet combined with GLPG2222 oral tablet and GLPG2737 oral capsule at up to 2 dose levels in ascending order.
GLPG3067/GLPG2222/GLPG2737 Placebo multiple dosePLACEBO_COMPARATORMultiple doses of GLPG3067 matching placebo oral tablet combined with GLPG2222 matching placebo oral tablet and GLPG2737 matching placebo oral capsule.
Interventions
NameTypeDescription
GLPG3067 single doseDRUGGLPG3067 oral suspension, single ascending doses, daily
Placebo single doseDRUGPlacebo, oral suspension, daily
GLPG3067 multiple doseDRUGGLPG3067 oral suspension, multiple ascending doses, daily for 14 days
Placebo multiple doseDRUGPlacebo, oral suspension, daily for 14 days
GLPG3067 oral suspensionDRUGGLPG3067 oral suspension, single dose, daily
GLPG3067 oral tabletDRUGGLPG3067 oral tablet, single dose, daily
GLPG3067/GLPG2222 multiple doseDRUGGLPG3067 oral suspension and GLPG2222 oral tablet, multiple doses, daily for 14 days
GLPG3067/GLPG2222 Placebo multiple doseDRUGGLPG3067 matching placebo oral suspension and GLPG2222 matching placebo oral tablet, multiple doses, daily for 14 days
GLPG3067/GLPG2222/GLPG2737 multiple doseDRUGGLPG3067 oral tablet, GLPG2222 oral tablet and GLPG2737 oral capsule, multiple doses, daily for 14 days
GLPG3067/GLPG2222/GLPG2737 Placebo multiple doseDRUGGLPG3067 matching placebo oral tablet, GLPG2222 matching placebo oral tablet and GLPG2737 matching placebo oral capsule, multiple doses, daily for 14 days
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Eligibility Criteria
Age Range18 Years — 70 Years
SexFEMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Female subject between 18-70 years of age, inclusive, on the date of signing the informed consent form (ICF). * Be of non-childbearing potential defined as surgically sterile (hysterectomy, bilateral salpingectomy and bilateral oophorectomy), or post-menopausal (at least 12 co...

Countries:Belgium
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