Recent Updates
Recently added Catalysts

GLPG1972

Phase 2

Osteoarthritis | Small molecule | Musculoskeletal |Galapagos NV|Last Updated: Jul 28, 2021

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
Premium
Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
Premium
Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLEDDMC
Total Trials1
Total Enrollment932
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT03595618A Study to Assess Efficacy and Safety of GLPG1972/S201086 in Participants With Knee OsteoarthritisPHASE2 COMPLETED 932Aug 14, 2018Jul 14, 2020Jul 28, 202144 United States
Unlock Drug Trial Details
Study Endpoints
Primary Endpoints
Change From Baseline in Cartilage Thickness of the cMTFC as Assessed by qMRI on the Target Knee to Week 52
Baseline, Week 52

Reduction in cartilage loss was assessed by cartilage thickness as measured in the medial cMTFC of the target knee using qMRI.

Secondary Endpoints
Number of Participants Who Were Osteoarthritis (OA) Structural Progressors Based on Cartilage Thickness in the cMTFC Assessed by qMRI on the Target Knee
Week 52
Change From Baseline in Western Ontario and McMaster Universities Osteoarthritis Index (WOMAC) Total Score and Subscales Scores for Pain, Function, and Stiffness to Week 52
Baseline, Week 52
Change From Baseline in Pain Assessment in the Target Knee as Measured by Visual Analog Scale (VAS) to Week 52
Baseline, Week 52
Unlock Study Endpoints
Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
GLPG1972 75 mgEXPERIMENTALParticipants received 1 film-coated tablet of GLPG1972 75 mg and 3 GLPG1972 matching placebo tablets, orally once daily for 52 weeks.
GLPG1972 150 mgEXPERIMENTALParticipants received 2 film-coated tablets of GLPG1972 75 mg (total dose 150 mg) and 2 GLPG1972 matching placebo tablets, orally once daily for 52 weeks.
GLPG1972 300 mgEXPERIMENTALParticipants received 4 film-coated tablets of GLPG1972 75 mg (total dose 300 mg), orally once daily for 52 weeks.
PlaceboPLACEBO_COMPARATORParticipants received 4 film-coated tablets of GLPG1972 matching placebo, orally once daily for 52 weeks.
Interventions
NameTypeDescription
GLPG1972DRUGFilm-coated tablets of GLPG1972 for oral use.
PlaceboDRUGFilm-coated tablets of matching placebo for oral use.
Unlock Study Design Details
Eligibility Criteria
Age Range40 Years — 75 Years
SexALL
Healthy VolunteersNo
Study Sites44

Inclusion Criteria: * Male participants or female participants of non-childbearing potential and not breastfeeding. * Body weight \> 40 kg, body mass index (BMI) \< 40 kg/m\^2. * Diagnosed for knee osteoarthritis based on clinical and radiological criteria of the American College of Rheumatology. *...

Countries:United States
Unlock Eligibility Criteria