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GLPG1205 single ascending doses,

Phase 1

Healthy | Small molecule | Other |Galapagos NV|Last Updated: Oct 16, 2013

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedDouble-BlindPLACEBO_CONTROLLED
Total Trials1
Total Enrollment40
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01887106First-in-Human Single and Multiple Dose of GLPG1205PHASE1 COMPLETED 40Jun 1, 2013Oct 1, 2013Oct 16, 20131 Belgium
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Study Endpoints
Primary Endpoints
Safety and tolerability after single dose
Between screening and 7-10 days after the last dose

To evaluate the safety and tolerability of GLPG1205 in comparison with placebo after a single oral dose in healthy subjects in terms of adverse events, physical examinations, vital signs, ECG and lab assessments

Safety and tolerability after multiple doses
Between screening and 7-10 days after the last dose

To evaluate the safety and tolerability of GLPG1205 in comparison with placebo after multiple oral doses daily for 14 days in healthy subjects in terms of adverse events, physical examinations, vital signs, ECG and lab assessments

Secondary Endpoints
The amount of GLPG1205 in plasma and urine over time after a single oral dose
Between Day 1 predose and 48 hours post dose
The amount of GLPG1205 in plasma and urine over time after multiple oral doses
Between Day 1 predose and Day 16 (48 hours after the last dose)
Ratio of 6-b-hydroxycortisol/cortisol in urine
Twelve hours before dosing on Day 1 and Day 14
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Study Design & Arms
AllocationRANDOMIZED
MaskingQUADRUPLE
ModelPARALLEL
PurposeTREATMENT
Treatment Arms
ArmTypeDescription
GLPG1205 single doseEXPERIMENTALSingle oral dose of GLPG1205 suspension - ascending doses
Placebo single dosePLACEBO_COMPARATORSingle oral dose of placebo suspension
GLPG1205 multiple dosesEXPERIMENTALMultiple oral doses of GLPG1205 suspension - ascending doses
Placebo multiple dosesPLACEBO_COMPARATORMultiple oral doses of placebo suspension
Interventions
NameTypeDescription
GLPG1205 single ascending doses, oral suspensionDRUGSingle dose, oral suspension at 10 mg/mL or 50 mg/mL, starting dose of 10mg escalating up to 800mg
Placebo single ascending doses, oral suspensionDRUGSingle dose, oral suspension matching placebo
GLPG1205, multiple ascending doses, oral suspensionDRUGMultiple doses, daily for 14 days, oral suspension at 10 mg/mL or 50 mg/mL, anticipated doses: 100mg to 400mg
Placebo, multiple ascending doses, oral suspensionDRUGMultiple doses, daily for 14 days, oral suspension matching placebo
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Eligibility Criteria
Age Range18 Years — 50 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male, age 18-50 years * BMI between 18-30 kg/m2 Exclusion Criteria: * Any condition that might interfere with the procedures or tests in this study * Drug or alcohol abuse * Smoking

Countries:Belgium
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