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GLPG1205 film-coated

Phase 1

Healthy | Small molecule | Other |Galapagos NV|Last Updated: Mar 25, 2021

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
CONTROLLEDBiomarker
Total Trials1
Total Enrollment12
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT04704739Evaluation of Mass Balance and Absolute Bioavailability of GLPG1205PHASE1 COMPLETED 12Jan 13, 2021Mar 10, 2021Mar 25, 20211 United Kingdom
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Study Endpoints
Primary Endpoints
Absolute oral bioavailability (F) (%)
Between Day 1 and Day 22

To determine the absolute bioavailability of an oral dose of GLPG1205 relative to an intravenous (i.v.) microtracer dose of \[14C\]-GLPG1205

Recovery of total radioactivity in urine and feces measured as amount of [14C]-GLPG1205 excreted as percentage of the administered dose (Ae%)
Between Day 1 and Day 22

To assess the mass balance recovery after a single oral dose of \[14C\]-GLPG1205

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Study Design & Arms
AllocationNON_RANDOMIZED
MaskingNONE
ModelSEQUENTIAL
PurposeBASIC_SCIENCE
Treatment Arms
ArmTypeDescription
GLPG1205 oral and [14C]-GLPG1205 IVEXPERIMENTALSingle oral dose of GLPG1205 followed by \[14C\]-GLPG1205 solution for infusion
[14C]-GLPG1205 capsuleEXPERIMENTALSingle oral dose of GLPG1205 as solid formulation
Interventions
NameTypeDescription
GLPG1205 film-coated tabletsDRUGSingle oral dose of GLPG1205
[14C]-GLPG1205 solution for infusionDRUGA 15-minute IV infusion of \[14C\]-GLPG1205
GLPG1205 capsulesDRUGSingle oral dose of GLPG1205 as solid formulation
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Eligibility Criteria
Age Range18 Years — 64 Years
SexMALE
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Male between 18-64 years of age (extremes included) (Part 1) and between 45-64 years of age (extremes included) (Part 2), on the date of signing the informed consent form. * A body mass index (BMI) between 18.0-32.0 kg/m2, inclusive. * Having a regular (at least) daily defecat...

Countries:United Kingdom
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