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ASA /esomeprazole

Phase 1

Healthy | Small molecule | Other |AstraZeneca PLC|Last Updated: May 10, 2012

Success Probability
Approval Probability 71%
TA Base Rate26%
Adjusted LOA41%
ML RiskLOW_RISK
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Market & Valuation
rNPV $3.2B
Market Size $9.4B
Revenue Basis $1.6B
Competitors 6
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Trial Design
RandomizedACTIVE_CONTROLLED
Total Trials1
Total Enrollment54
FDA Designations
No designations recorded
Clinical Trials (1)
NCT IDTitlePhaseStatusEnrollmentVelocityDesignStartCompletionLast UpdatedSitesCountries
NCT01448031A Healthy Female and Male Volunteers Aspirin StudyPHASE1 COMPLETED 54Nov 1, 2011Apr 1, 2012May 10, 20121 United Kingdom
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Study Endpoints
Primary Endpoints
pharmacokinetic profile of acetylsalicylic acid (ASA) and salicylic acid (SA) in terms of area under curve (AUC), maximum concentration at steady state (Css,max), time to reach maximum concentration (tmax) and terminal half- time (t1/2).
Day 5

PK samples collected pre-dose and at 5mins, 10 mins, 20 mins, 30 mins, 40mins, 50 mins, 1hr 15 mins, 1.5hrs, 2 hrs, 2hr 30 mins, 3hrs, 3hr 30 mins, 4 hrs, 5 hrs, 6hrs, 8hrs,10 hrs, 12hrs post-dose.

Secondary Endpoints
Description of the safety profile in terms of adverse events, blood pressure, pulse, ECG (Electrocardiogram), physical examination, safety labs
Pre-dose up to 7 day after last dose
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Study Design & Arms
AllocationRANDOMIZED
MaskingNONE
ModelCROSSOVER
PurposeDIAGNOSTIC
Treatment Arms
ArmTypeDescription
1EXPERIMENTALCapsule ASA 81mg/esomeprazole 20mg
2ACTIVE_COMPARATORASA (Acetylsalicylzuur Apotex cardio 80 mg) Tablet 80 mg
Interventions
NameTypeDescription
Capsule ASA 81mg/esomeprazole 20mgDRUGMultiple doses administered on Day 1 to 5
Acetylsalicylzuur Apotex CardioDRUGMultiple doses administered on Day 1 to 5
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Eligibility Criteria
Age Range20 Years — 50 Years
SexALL
Healthy VolunteersYes
Study Sites1

Inclusion Criteria: * Healthy male and female subjects aged 20 to 50 years inclusive. * Have a body body mass index (BMI) of 18.0 to 30.0 kg/m2 inclusive and weigh 50.0 to 100.0 kg inclusive. * Females must be of non-childbearing potential or be of childbearing potential but have a negative serum h...

Countries:United Kingdom
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